#------------------------------------------------------------------------------ #$Date: 2025-08-18 23:52:38 +0100 (Mon, 18 Aug 2025) $ #$Revision: 301791 $ #$URL: svn://www.crystallography.net/cod/cif/2/00/52/2005252.cif $ #------------------------------------------------------------------------------ # # This file is available in the Crystallography Open Database (COD), # http://www.crystallography.net/. The original data for this entry # were provided by IUCr Journals, http://journals.iucr.org/. # # The file may be used within the scientific community so long as # proper attribution is given to the journal article from which the # data were obtained. # data_2005252 loop_ _publ_author_name 'Sch\"afer, M.' 'Herbst-Irmer, R.' 'Pohl, E.' 'Sch\"unke, C.' 'Tietze, L. F.' _publ_section_title ;(2R)-3-[(4S)-4-Benzyl-2-oxo-3-oxazolidinyl]-3-oxo-2-[(1R,2S)-2-vinylcyclohexyl]propionic Acid Methyl Ester and (2R)-3-[(4S)-4-Benzyl-2-oxo-3-oxazolidinyl]-3-oxo-2-[(1R,2S)-2-vinylcyclopentyl]propionic Acid Methyl Ester ; _journal_issue 8 _journal_name_full 'Acta Crystallographica Section C' _journal_page_first 2029 _journal_page_last 2032 _journal_paper_doi 10.1107/S010827019600159X _journal_volume 52 _journal_year 1996 _chemical_formula_sum 'C22 H27 N O5' _chemical_formula_weight 385.45 _chemical_name_systematic ; (1'R,2R,2'S,4"S)-3-(4"-Benzyl-oxazolidin-2"-one-3"-yl) -3-oxo-2-(2'-vinyl-cyclohexyl)-propionic acid methyl ester ; _space_group_IT_number 19 _symmetry_cell_setting orthorhombic _symmetry_space_group_name_Hall 'P 2ac 2ab' _symmetry_space_group_name_H-M 'P 21 21 21' _audit_creation_method SHELXL _cell_angle_alpha 90 _cell_angle_beta 90 _cell_angle_gamma 90 _cell_formula_units_Z 4 _cell_length_a 9.3870(4) _cell_length_b 10.0616(4) _cell_length_c 21.722(1) _cell_measurement_reflns_used 75 _cell_measurement_temperature 293(2) _cell_measurement_theta_max 28 _cell_measurement_theta_min 10.5 _cell_volume 2051.60(15) _computing_cell_refinement XSCANS _computing_data_collection 'XSCANS (Siemens, 1994)' _computing_data_reduction XSCANS _computing_molecular_graphics 'SHELXTL-Plus (Sheldrick, 1994)' _computing_publication_material SHELXL93 _computing_structure_refinement 'SHELXL93 (Sheldrick, 1993)' _computing_structure_solution 'SHELXS86 (Sheldrick, 1990)' _diffrn_ambient_temperature 293(2) _diffrn_measurement_device 'Siemens P4 four-circle diffractometer' _diffrn_measurement_method 'profile from \q/2\q' _diffrn_radiation_monochromator graphite _diffrn_radiation_source 'fine-focus sealed tube' _diffrn_radiation_type CuK\a _diffrn_radiation_wavelength 1.54178 _diffrn_reflns_av_R_equivalents 0.0504 _diffrn_reflns_av_sigmaI/netI 0.0456 _diffrn_reflns_limit_h_max 10 _diffrn_reflns_limit_h_min -10 _diffrn_reflns_limit_k_max 10 _diffrn_reflns_limit_k_min -10 _diffrn_reflns_limit_l_max 23 _diffrn_reflns_limit_l_min -23 _diffrn_reflns_number 5345 _diffrn_reflns_theta_max 56.74 _diffrn_reflns_theta_min 4.07 _diffrn_standards_decay_% 0 _diffrn_standards_interval_count 100 _diffrn_standards_number 3 _exptl_absorpt_coefficient_mu 0.719 _exptl_absorpt_correction_type none _exptl_crystal_colour colourless _exptl_crystal_density_diffrn 1.248 _exptl_crystal_density_method none _exptl_crystal_description block _exptl_crystal_F_000 824 _exptl_crystal_size_max 0.5 _exptl_crystal_size_mid 0.4 _exptl_crystal_size_min 0.4 _refine_diff_density_max .163 _refine_diff_density_min -.129 _refine_ls_abs_structure_details 'Flack (1983)' _refine_ls_abs_structure_Flack -0.0(3) _refine_ls_extinction_coef 0.0060(6) _refine_ls_extinction_method 'SHELXL93 (Sheldrick, 1993)' _refine_ls_goodness_of_fit_all 1.044 _refine_ls_goodness_of_fit_obs 1.064 _refine_ls_hydrogen_treatment 'H atoms riding' _refine_ls_matrix_type full _refine_ls_number_parameters 255 _refine_ls_number_reflns 2731 _refine_ls_number_restraints 0 _refine_ls_restrained_S_all 1.044 _refine_ls_restrained_S_obs 1.064 _refine_ls_R_factor_all 0.0491 _refine_ls_R_factor_obs 0.0429 _refine_ls_shift/esd_max 0.000 _refine_ls_shift/esd_mean 0.000 _refine_ls_structure_factor_coef Fsqd _refine_ls_weighting_details 'w = 1/[\s^2^(Fo^2^)+(0.0715P)^2^+0.0545P] where P=(Fo^2^+2Fc^2^)/3' _refine_ls_weighting_scheme calc _refine_ls_wR_factor_all 0.1122 _refine_ls_wR_factor_obs 0.1072 _reflns_number_observed 2428 _reflns_number_total 2732 _reflns_observed_criterion >2sigma(I) _cod_data_source_file jz1097.cif _cod_data_source_block I _cod_depositor_comments ; The following automatic conversions were performed: '_refine_ls_weighting_scheme' value 'calc w = 1/[\s^2^(Fo^2^)+(0.0715P)^2^+0.0545P] where P=(Fo^2^+2Fc^2^)/3' was changed to 'calc'. New tag '_refine_ls_weighting_details' was created. The value of the new tag was set to 'w = 1/[\s^2^(Fo^2^)+(0.0715P)^2^+0.0545P] where P=(Fo^2^+2Fc^2^)/3'. Automatic conversion script Id: cif_fix_values 3143 2015-03-26 13:38:13Z robertas ; _cod_original_cell_volume 2051.6(2) _cod_database_code 2005252 loop_ _symmetry_equiv_pos_as_xyz 'x, y, z' '-x+1/2, -y, z+1/2' '-x, y+1/2, -z+1/2' 'x+1/2, -y+1/2, -z' loop_ _atom_site_aniso_label _atom_site_aniso_U_11 _atom_site_aniso_U_22 _atom_site_aniso_U_33 _atom_site_aniso_U_12 _atom_site_aniso_U_13 _atom_site_aniso_U_23 O1 0.190(3) 0.0872(15) 0.0585(12) -0.0361(19) 0.0367(15) -0.0044(12) C2 0.105(2) 0.072(2) 0.0577(16) -0.012(2) 0.0199(16) -0.0017(15) O2 0.153(2) 0.0637(13) 0.0649(12) -0.0100(15) 0.0192(14) 0.0036(10) N3 0.0760(14) 0.0554(12) 0.0513(12) -0.0084(12) 0.0106(11) -0.0031(10) C4 0.0730(18) 0.0665(16) 0.0564(15) -0.0107(15) 0.0142(14) -0.0121(12) C5 0.169(4) 0.095(2) 0.078(2) -0.044(3) 0.050(2) -0.0235(19) C1' 0.0465(14) 0.0521(14) 0.0577(13) 0.0005(12) 0.0024(12) -0.0004(11) O3 0.0849(13) 0.0535(11) 0.0639(11) 0.0051(10) 0.0034(10) -0.0037(8) C2' 0.0396(11) 0.0453(12) 0.0566(12) 0.0015(11) 0.0017(10) -0.0013(11) C3' 0.0434(14) 0.0594(15) 0.0617(14) -0.0049(12) 0.0032(12) -0.0001(12) O4 0.0473(10) 0.1056(15) 0.1110(16) -0.0045(12) 0.0212(11) -0.0294(14) O5 0.0487(10) 0.0604(10) 0.0815(11) -0.0154(9) 0.0019(9) -0.0046(9) C4' 0.0579(16) 0.092(2) 0.091(2) -0.0319(17) -0.0035(15) 0.0023(18) C1'' 0.0375(11) 0.0461(12) 0.0532(13) 0.0003(10) 0.0015(10) -0.0027(11) C2'' 0.0422(12) 0.0488(12) 0.0595(13) -0.0028(11) 0.0030(11) 0.0002(12) C3'' 0.0543(15) 0.0624(15) 0.0709(15) -0.0059(14) 0.0167(13) -0.0019(14) C4'' 0.0728(18) 0.0723(17) 0.0523(13) -0.0040(15) 0.0087(13) 0.0029(14) C5'' 0.0683(17) 0.0753(17) 0.0592(14) -0.0025(16) -0.0067(14) 0.0050(13) C6'' 0.0442(13) 0.0645(15) 0.0610(14) 0.0008(13) -0.0029(12) 0.0068(13) C7'' 0.0390(13) 0.0786(19) 0.090(2) -0.0009(13) -0.0005(14) 0.0201(17) C8'' 0.0589(18) 0.141(3) 0.094(2) -0.007(2) -0.0181(17) 0.028(2) C41 0.0605(17) 0.0752(17) 0.0642(15) 0.0023(15) 0.0008(13) -0.0108(14) C42 0.0517(14) 0.0636(15) 0.0522(13) -0.0052(14) 0.0023(12) 0.0020(13) C43 0.0522(15) 0.0698(17) 0.0686(16) 0.0021(15) -0.0048(13) -0.0012(14) C44 0.0617(17) 0.087(2) 0.0667(16) -0.0047(17) -0.0112(13) -0.0103(17) C45 0.0666(18) 0.0703(17) 0.0735(17) -0.0075(17) 0.0043(15) -0.0113(15) C46 0.0752(19) 0.0623(17) 0.0751(18) 0.0023(15) -0.0008(16) 0.0031(15) C47 0.0722(17) 0.0727(18) 0.0536(13) -0.0015(16) -0.0104(12) 0.0096(13) loop_ _atom_site_label _atom_site_occupancy _atom_site_fract_x _atom_site_fract_y _atom_site_fract_z _atom_site_U_iso_or_equiv _atom_site_thermal_displace_type _atom_site_calc_flag _atom_site_refinement_flags _atom_site_type_symbol O1 1 .1978(3) .7417(2) -.01621(9) .112(1) Uani d . O C2 1 .1819(4) .7641(3) .0437(1) .0783(9) Uani d . C O2 1 .1849(3) .8742(2) .06487(9) .0938(8) Uani d . O N3 1 .1598(3) .6447(2) .07385(9) .0609(6) Uani d . N C4 1 .1575(3) .5323(3) .0301(1) .0653(7) Uani d . C H4 1 .228 .4654 .0422 .078 Uiso calc R H C5 1 .2048(5) .6018(4) -.0287(2) .114(2) Uani d . C H5A 1 .3012 .5761 -0.0394 .137 Uiso calc R H H5B 1 .1421 .579(7) -0.0626 .137 Uiso calc R H C1' 1 .1648(3) .6227(3) .1369(1) .0521(6) Uani d . C O3 1 .1636(2) .5086(2) .15593(7) .0674(5) Uani d . O C2' 1 .1688(2) .7435(2) .1790(1) .0472(5) Uani d . C H2' 1 .1064 .8114 .1612 .057 Uiso calc R H C3' 1 .3205(3) .7971(2) .1779(1) .0548(6) Uani d . C O4 1 .4202(2) .7443(3) .1542(1) .0879(7) Uani d . O O5 1 .3285(2) .9088(2) .21004(8) .0636(5) Uani d . O C4' 1 .4693(3) .9637(3) .2194(2) .0805(9) Uani d . C H4'A 1 .4621 1.0447 .2425 .121 Uiso calc R H H4'B 1 .5124 .982(5) .1802 .121 Uiso calc R H H4'C 1 .5268 .9011 .2416 .121 Uiso calc R H C1'' 1 .1210(2) .7199(2) .2461(1) .0456(6) Uani d . C H1'' 1 .1082 .8086 .264 .055 Uiso calc R H C2'' 1 -.0241(2) .6504(2) .2528(1) .0501(6) Uani d . C H2'' 1 -0.0136 .5585 .2384 .06 Uiso calc R H C3'' 1 -.0662(3) .6465(3) .3210(1) .0625(7) Uani d . C H3''A 1 -0.0827 .7366 .3352 .075 Uiso calc R H H3''B 1 -0.1547 .598(5) .3253 .075 Uiso calc R H C4'' 1 .0473(3) .5819(3) .3613(1) .0658(7) Uani d . C H4''D 1 .0182 .5865 .4041 .079 Uiso calc R H H4''E 1 .057 .489(5) .3502 .079 Uiso calc R H C5'' 1 .1889(3) .6514(3) .3534(1) .0676(7) Uani d . C H5''A 1 .2609 .6062 .3777 .081 Uiso calc R H H5''B 1 .1815 .742(5) .3682 .081 Uiso calc R H C6'' 1 .2328(3) .6518(3) .2861(1) .0565(6) Uani d . C H6''A 1 .2458 .5611 .2721 .068 Uiso calc R H H6''B 1 .323 .698(4) .2817 .068 Uiso calc R H C7'' 1 -0.1377(3) .7147(3) .2154(1) .0693(8) Uani d . C H7'' 1 -0.1588 .8028 .2245 .083 Uiso calc R H C8'' 1 -0.2104(3) .6592(5) .1712(2) .098(1) Uani d . C H8''A 1 -0.1931 .5712 .1605 .117 Uiso calc R H H8''B 1 -0.2797 .708(7) .1504 .117 Uiso calc R H C41 1 .0107(3) .4694(3) .0255(1) .0666(7) Uani d . C H41A 1 -0.0199 .4415 .0662 .08 Uiso calc R H H41B 1 -0.0566 .535(5) .0107 .08 Uiso calc R H C42 1 .0096(3) .3510(3) -.0173(1) .0558(6) Uani d . C C43 1 -.0728(3) .3487(3) -.0705(1) .0635(7) Uani d . C H43 1 -0.1274 .4225 -0.0809 .076 Uiso calc R H C44 1 -.0743(3) .2382(3) -0.1080(1) .0718(8) Uani d . C H44 1 -0.1292 .2385 -0.1436 .086 Uiso calc R H C45 1 .0039(3) .1287(3) -.0933(1) .0702(8) Uani d . C H45 1 .0018 .0542 -0.1186 .084 Uiso calc R H C46 1 .0852(3) .1287(3) -.0414(1) .0708(8) Uani d . C H46 1 .1388 .0541 -0.0312 .085 Uiso calc R H C47 1 .0881(3) .2395(3) -.0037(1) .0662(7) Uani d . C H47 1 .1443 .2385 .0315 .079 Uiso calc R H loop_ _atom_type_symbol _atom_type_description _atom_type_scat_dispersion_real _atom_type_scat_dispersion_imag _atom_type_scat_source C C .0181 .0091 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' H H .0000 .0000 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' N N .0311 .0180 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' O O .0492 .0322 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' loop_ _geom_angle_atom_site_label_1 _geom_angle_atom_site_label_2 _geom_angle_atom_site_label_3 _geom_angle _geom_angle_publ_flag C2 O1 C5 110.9(2) y O2 C2 O1 122.0(3) y O2 C2 N3 128.5(2) y O1 C2 N3 109.5(3) y C2 N3 C1' 126.9(2) y C2 N3 C4 111.2(2) y C1' N3 C4 120.9(2) y N3 C4 C41 112.0(2) y N3 C4 C5 100.6(2) y C41 C4 C5 113.6(3) y O1 C5 C4 106.1(2) y O3 C1' N3 118.9(2) y O3 C1' C2' 123.3(2) y N3 C1' C2' 117.8(2) y C1' C2' C3' 107.30(19) y C1' C2' C1'' 115.94(19) y C3' C2' C1'' 109.91(19) y O4 C3' O5 124.1(2) y O4 C3' C2' 125.6(2) y O5 C3' C2' 110.2(2) y C3' O5 C4' 116.7(2) y C6'' C1'' C2'' 110.64(19) ? C6'' C1'' C2' 113.98(19) ? C2'' C1'' C2' 114.56(18) ? C7'' C2'' C3'' 110.7(2) ? C7'' C2'' C1'' 112.70(19) ? C3'' C2'' C1'' 109.27(19) ? C4'' C3'' C2'' 112.7(2) ? C5'' C4'' C3'' 110.6(2) ? C4'' C5'' C6'' 110.5(2) ? C5'' C6'' C1'' 111.2(2) ? C8'' C7'' C2'' 126.2(3) ? C42 C41 C4 112.0(2) ? C47 C42 C43 117.6(3) ? C47 C42 C41 120.6(2) ? C43 C42 C41 121.9(3) ? C44 C43 C42 120.7(3) ? C45 C44 C43 120.5(3) ? C46 C45 C44 119.7(3) ? C45 C46 C47 120.1(3) ? C42 C47 C46 121.4(2) ? loop_ _geom_bond_atom_site_label_1 _geom_bond_atom_site_label_2 _geom_bond_distance _geom_bond_publ_flag O1 C2 1.328(3) y O1 C5 1.434(4) y C2 O2 1.201(4) y C2 N3 1.385(4) y N3 C1' 1.388(3) y N3 C4 1.477(3) y C4 C41 1.520(4) ? C4 C5 1.523(4) y C1' O3 1.221(3) y C1' C2' 1.521(3) y C2' C3' 1.523(3) y C2' C1'' 1.545(3) y C3' O4 1.192(3) y C3' O5 1.325(3) y O5 C4' 1.447(3) y C1'' C6'' 1.524(3) ? C1'' C2'' 1.538(3) ? C2'' C7'' 1.488(4) ? C2'' C3'' 1.534(4) ? C3'' C4'' 1.525(4) ? C4'' C5'' 1.511(4) ? C5'' C6'' 1.521(4) ? C7'' C8'' 1.304(4) y C41 C42 1.512(4) ? C42 C47 1.374(4) ? C42 C43 1.391(4) ? C43 C44 1.378(4) ? C44 C45 1.363(4) ? C45 C46 1.361(4) ? C46 C47 1.384(4) ? loop_ _cod_related_entry_id _cod_related_entry_database _cod_related_entry_code 1 ChemSpider 10265491 2 PubChem 21633694