#------------------------------------------------------------------------------ #$Date: 2025-08-19 11:43:10 +0100 (Tue, 19 Aug 2025) $ #$Revision: 301803 $ #$URL: svn://www.crystallography.net/cod/cif/2/20/45/2204560.cif $ #------------------------------------------------------------------------------ # # This file is available in the Crystallography Open Database (COD), # http://www.crystallography.net/. The original data for this entry # were provided by IUCr Journals, http://journals.iucr.org/. # # The file may be used within the scientific community so long as # proper attribution is given to the journal article from which the # data were obtained. # data_2204560 loop_ _publ_author_name 'Ameijde, Jeroen van' 'Cowley, Andrew R.' 'Fleet, George W. J.' 'Nash, Robert J.' 'Iezzi Simone, Michela' 'Soengas, Raquel' _publ_section_title 5-Amino-5-deoxy-2-C-hydroxymethyl-2,3-O-isopropylidene-D-talono-1,5-lactam _journal_issue 11 _journal_name_full 'Acta Crystallographica Section E' _journal_page_first o2140 _journal_page_last o2141 _journal_paper_doi 10.1107/S1600536804025292 _journal_volume 60 _journal_year 2004 _chemical_formula_iupac 'C10 H17 N1 O6' _chemical_formula_moiety 'C10 H17 N1 O6' _chemical_formula_sum 'C10 H17 N O6' _chemical_formula_weight 247.25 _chemical_name_systematic ; 5-Amino-5-deoxy-2-C-hydroxymethyl-2,3-O-isopropylidene-D-talono-1,5-lactam ; _space_group_IT_number 4 _symmetry_cell_setting monoclinic _symmetry_space_group_name_Hall 'P 2yb' _symmetry_space_group_name_H-M 'P 1 21 1' _atom_sites_solution_hydrogens geom _atom_sites_solution_primary direct _cell_angle_alpha 90 _cell_angle_beta 99.6456(14) _cell_angle_gamma 90 _cell_formula_units_Z 2 _cell_length_a 6.1266(2) _cell_length_b 6.7254(2) _cell_length_c 13.8419(5) _cell_measurement_reflns_used 5291 _cell_measurement_temperature 150 _cell_measurement_theta_max 28 _cell_measurement_theta_min 5 _cell_volume 562.28(3) _computing_cell_refinement 'COLLECT and DENZO' _computing_data_collection 'COLLECT (Nonius, 2000)' _computing_data_reduction 'COLLECT and DENZO (Otwinowski & Minor, 1996)' _computing_molecular_graphics 'ATOMS (Shape Software, 2002)' _computing_publication_material CRYSTALS _computing_structure_refinement 'CRYSTALS (Betteridge et al., 2003)' _computing_structure_solution 'SIR92 (Altomare et al., 1994)' _diffrn_ambient_temperature 150 _diffrn_measured_fraction_theta_full 0.996 _diffrn_measured_fraction_theta_max 0.996 _diffrn_measurement_device_type 'Nonius KappaCCD' _diffrn_measurement_method \w _diffrn_radiation_monochromator graphite _diffrn_radiation_type MoK\a _diffrn_radiation_wavelength 0.71073 _diffrn_reflns_av_R_equivalents 0.030 _diffrn_reflns_limit_h_max 7 _diffrn_reflns_limit_h_min -7 _diffrn_reflns_limit_k_max 8 _diffrn_reflns_limit_k_min -8 _diffrn_reflns_limit_l_max 17 _diffrn_reflns_limit_l_min -17 _diffrn_reflns_number 5291 _diffrn_reflns_theta_full 27.425 _diffrn_reflns_theta_max 27.425 _diffrn_reflns_theta_min 5.112 _diffrn_standards_decay_% 0.00 _diffrn_standards_interval_count 0 _diffrn_standards_interval_time 0 _diffrn_standards_number 0 _exptl_absorpt_coefficient_mu 0.121 _exptl_absorpt_correction_T_max 0.98 _exptl_absorpt_correction_T_min 0.96 _exptl_absorpt_correction_type multi-scan _exptl_absorpt_process_details '(DENZO/SCALEPACK; Otwinowski & Minor, 1996)' _exptl_crystal_colour colourless _exptl_crystal_density_diffrn 1.460 _exptl_crystal_density_meas ? _exptl_crystal_description plate _exptl_crystal_F_000 264 _exptl_crystal_size_max 0.38 _exptl_crystal_size_mid 0.38 _exptl_crystal_size_min 0.14 _refine_diff_density_max 0.20 _refine_diff_density_min -0.16 _refine_ls_extinction_method None _refine_ls_goodness_of_fit_ref 1.0968 _refine_ls_hydrogen_treatment mixed _refine_ls_matrix_type full _refine_ls_number_parameters 170 _refine_ls_number_reflns 1211 _refine_ls_number_restraints 1 _refine_ls_R_factor_all 0.0334 _refine_ls_R_factor_gt 0.0276 _refine_ls_shift/su_max 0.003461 _refine_ls_structure_factor_coef F _refine_ls_weighting_details ; Method, part 1, Chebychev polynomial, (Watkin, 1994, Prince, 1982) [weight] = 1.0/[A~0~*T~0~(x)+A~1~*T~1~(x) ... +A~n-1~]*T~n-1~(x)] where A~i~ are the Chebychev coefficients listed below and x= Fcalc/Fmax Method = Robust Weighting (Prince, 1982) W = [weight] * [1-(deltaF/6*sigmaF)^2^]^2^ A~i~ are: 1.14 0.561 0.916 ; _refine_ls_weighting_scheme calc _refine_ls_wR_factor_all 0.0352 _refine_ls_wR_factor_gt 0.0343 _refine_ls_wR_factor_ref 0.0343 _reflns_number_gt 1211 _reflns_number_total 1372 _reflns_threshold_expression I>3.00u(I) _cod_data_source_file rz6003.cif _cod_data_source_block 4 _cod_depositor_comments ; The following automatic conversions were performed: '_exptl_crystal_density_meas' value 'none' was changed to '?' - the value is perceived as not measured. Automatic conversion script Id: cif_fix_values 3008 2015-01-20 13:52:24Z robertas ; _cod_original_sg_symbol_H-M 'P 21' _cod_original_formula_sum 'C10 H17 N1 O6' _cod_database_code 2204560 loop_ _symmetry_equiv_pos_as_xyz x,y,z -x,y+1/2,-z loop_ _atom_site_label _atom_site_fract_x _atom_site_fract_y _atom_site_fract_z _atom_site_U_iso_or_equiv _atom_site_adp_type _atom_site_occupancy _atom_site_type_symbol N1 0.1580(2) 0.3518(2) 0.37174(11) 0.0176 Uani 1.0000 N C1 0.1315(2) 0.2536(3) 0.28694(12) 0.0160 Uani 1.0000 C C2 0.3054(3) 0.2808(2) 0.21935(13) 0.0154 Uani 1.0000 C C3 0.4612(2) 0.4553(3) 0.24723(10) 0.0153 Uani 1.0000 C C4 0.5232(2) 0.4908(2) 0.35601(11) 0.0151 Uani 1.0000 C C5 0.3214(2) 0.5061(3) 0.40842(11) 0.0161 Uani 1.0000 C O1 -0.0245(2) 0.1385(2) 0.26071(10) 0.0239 Uani 1.0000 O C6 0.4241(3) 0.0847(3) 0.20754(13) 0.0206 Uani 1.0000 C O2 0.5652(2) 0.0291(2) 0.29613(10) 0.0215 Uani 1.0000 O O3 0.1949(2) 0.3367(2) 0.12375(9) 0.0211 Uani 1.0000 O O4 0.3350(2) 0.6200(2) 0.20346(9) 0.0182 Uani 1.0000 O C7 0.1964(3) 0.5502(3) 0.11614(12) 0.0183 Uani 1.0000 C C8 0.2954(3) 0.6069(3) 0.02649(14) 0.0292 Uani 1.0000 C C9 -0.0325(3) 0.6348(3) 0.11512(15) 0.0303 Uani 1.0000 C O5 0.66148(19) 0.66075(19) 0.37549(9) 0.0196 Uani 1.0000 O C10 0.2106(3) 0.7109(3) 0.40523(12) 0.0203 Uani 1.0000 C O6 0.0666(2) 0.7158(2) 0.47624(9) 0.0245 Uani 1.0000 O H1 0.050(5) 0.324(5) 0.411(2) 0.042(8) Uiso 1.0000 H H2 0.699(6) 0.064(6) 0.293(2) 0.054(9) Uiso 1.0000 H H3 0.604(6) 0.768(6) 0.340(2) 0.052(9) Uiso 1.0000 H H4 -0.075(5) 0.680(5) 0.4463(19) 0.038(7) Uiso 1.0000 H H31 0.6060 0.4317 0.2249 0.0186 Uiso 1.0000 H H41 0.6082 0.3709 0.3835 0.0179 Uiso 1.0000 H H51 0.3818 0.4842 0.4793 0.0194 Uiso 1.0000 H H61 0.5153 0.0999 0.1545 0.0252 Uiso 1.0000 H H62 0.3111 -0.0220 0.1891 0.0252 Uiso 1.0000 H H81 0.2976 0.7550 0.0203 0.0355 Uiso 1.0000 H H82 0.4501 0.5545 0.0336 0.0355 Uiso 1.0000 H H83 0.2039 0.5485 -0.0334 0.0355 Uiso 1.0000 H H91 -0.0270 0.7829 0.1098 0.0358 Uiso 1.0000 H H92 -0.0858 0.5974 0.1771 0.0358 Uiso 1.0000 H H93 -0.1361 0.5800 0.0578 0.0358 Uiso 1.0000 H H101 0.3263 0.8163 0.4205 0.0247 Uiso 1.0000 H H102 0.1232 0.7347 0.3385 0.0247 Uiso 1.0000 H loop_ _atom_site_aniso_label _atom_site_aniso_U_11 _atom_site_aniso_U_22 _atom_site_aniso_U_33 _atom_site_aniso_U_12 _atom_site_aniso_U_13 _atom_site_aniso_U_23 N1 0.0164(7) 0.0179(7) 0.0198(6) -0.0030(5) 0.0066(5) 0.0004(6) C1 0.0130(7) 0.0138(7) 0.0217(8) 0.0014(6) 0.0043(5) 0.0041(6) C2 0.0166(7) 0.0140(7) 0.0159(8) -0.0015(6) 0.0038(6) 0.0003(6) C3 0.0151(6) 0.0147(7) 0.0167(7) -0.0016(6) 0.0045(5) 0.0009(6) C4 0.0140(7) 0.0152(8) 0.0155(7) -0.0008(5) 0.0011(5) -0.0004(6) C5 0.0147(7) 0.0186(7) 0.0152(7) -0.0019(6) 0.0026(5) -0.0004(6) O1 0.0182(6) 0.0233(6) 0.0307(6) -0.0075(5) 0.0056(4) -0.0016(6) C6 0.0246(8) 0.0146(8) 0.0237(9) 0.0000(6) 0.0076(6) -0.0018(6) O2 0.0155(6) 0.0166(6) 0.0326(7) -0.0008(5) 0.0047(5) 0.0034(5) O3 0.0300(7) 0.0156(6) 0.0166(6) -0.0047(5) 0.0004(5) -0.0006(5) O4 0.0234(6) 0.0134(5) 0.0162(6) -0.0013(4) -0.0010(4) 0.0009(4) C7 0.0208(8) 0.0164(8) 0.0170(8) -0.0048(6) 0.0011(6) 0.0010(6) C8 0.0362(10) 0.0332(11) 0.0192(8) -0.0112(9) 0.0076(7) 0.0018(7) C9 0.0208(9) 0.0315(10) 0.0371(10) 0.0010(8) 0.0004(7) 0.0023(9) O5 0.0141(5) 0.0185(6) 0.0248(6) -0.0042(5) -0.0007(4) -0.0012(5) C10 0.0178(7) 0.0227(8) 0.0213(8) -0.0004(6) 0.0063(6) -0.0046(7) O6 0.0161(5) 0.0370(7) 0.0215(6) -0.0008(5) 0.0060(4) -0.0103(6) loop_ _atom_type_symbol _atom_type_scat_dispersion_real _atom_type_scat_dispersion_imag _atom_type_scat_source 'C ' 0.0033 0.0016 International_Tables_Vol_IV_Table_2.2B 'H ' 0.0000 0.0000 International_Tables_Vol_IV_Table_2.2B 'N ' 0.0061 0.0033 International_Tables_Vol_IV_Table_2.2B 'O ' 0.0106 0.0060 International_Tables_Vol_IV_Table_2.2B loop_ _geom_angle_atom_site_label_1 _geom_angle_atom_site_label_2 _geom_angle_atom_site_label_3 _geom_angle _geom_angle_publ_flag C1 N1 C5 128.95(13) no C1 N1 H1 114.5(19) no C5 N1 H1 116.(2) no N1 C1 C2 118.74(14) no N1 C1 O1 122.89(15) no C2 C1 O1 118.36(15) no C1 C2 C3 113.93(13) no C1 C2 C6 110.60(13) no C3 C2 C6 113.79(13) no C1 C2 O3 108.93(13) no C3 C2 O3 102.22(13) no C6 C2 O3 106.70(13) no C2 C3 C4 114.70(13) no C2 C3 O4 102.65(12) no C4 C3 O4 109.21(13) no C2 C3 H31 110.567 no C4 C3 H31 104.177 no O4 C3 H31 115.933 no C3 C4 C5 113.15(13) no C3 C4 O5 111.05(13) no C5 C4 O5 110.94(13) no C3 C4 H41 106.285 no C5 C4 H41 106.403 no O5 C4 H41 108.711 no N1 C5 C4 110.13(13) no N1 C5 C10 110.58(13) no C4 C5 C10 115.68(13) no N1 C5 H51 110.696 no C4 C5 H51 104.970 no C10 C5 H51 104.465 no C2 C6 O2 111.42(13) no C2 C6 H61 108.982 no O2 C6 H61 108.982 no C2 C6 H62 108.982 no O2 C6 H62 108.982 no H61 C6 H62 109.467 no C6 O2 H2 109(2) no C2 O3 C7 108.74(13) no C3 O4 C7 107.81(13) no O3 C7 O4 105.95(14) no O3 C7 C8 108.57(16) no O4 C7 C8 110.19(14) no O3 C7 C9 111.03(15) no O4 C7 C9 107.58(15) no C8 C7 C9 113.27(16) no C7 C8 H81 109.467 no C7 C8 H82 109.467 no H81 C8 H82 109.476 no C7 C8 H83 109.467 no H81 C8 H83 109.476 no H82 C8 H83 109.476 no C7 C9 H91 109.467 no C7 C9 H92 109.467 no H91 C9 H92 109.476 no C7 C9 H93 109.467 no H91 C9 H93 109.476 no H92 C9 H93 109.476 no C4 O5 H3 112(2) no C5 C10 O6 108.81(14) no C5 C10 H101 109.637 no O6 C10 H101 109.637 no C5 C10 H102 109.637 no O6 C10 H102 109.637 no H101 C10 H102 109.467 no C10 O6 H4 109.0(16) no loop_ _geom_bond_atom_site_label_1 _geom_bond_atom_site_label_2 _geom_bond_distance _geom_bond_publ_flag N1 C1 1.333(2) no N1 C5 1.471(2) no N1 H1 0.94(3) no C1 C2 1.542(2) no C1 O1 1.236(2) no C2 C3 1.521(2) no C2 C6 1.528(2) no C2 O3 1.432(2) no C3 C4 1.509(2) no C3 O4 1.426(2) no C3 H31 1.000 no C4 C5 1.538(2) no C4 O5 1.4215(19) no C4 H41 1.000 no C5 C10 1.533(2) no C5 H51 1.000 no C6 O2 1.427(2) no C6 H61 1.000 no C6 H62 1.000 no O2 H2 0.86(3) no O3 C7 1.440(2) no O4 C7 1.435(2) no C7 C8 1.518(2) no C7 C9 1.511(2) no C8 H81 1.000 no C8 H82 1.000 no C8 H83 1.000 no C9 H91 1.000 no C9 H92 1.000 no C9 H93 1.000 no O5 H3 0.91(4) no C10 O6 1.427(2) no C10 H101 1.000 no C10 H102 1.000 no O6 H4 0.93(3) no loop_ _geom_hbond_atom_site_label_D _geom_hbond_atom_site_label_H _geom_hbond_atom_site_label_A _geom_hbond_site_symmetry_A _geom_hbond_distance_DH _geom_hbond_distance_HA _geom_hbond_distance_DA _geom_hbond_angle_DHA _geom_hbond_publ_flag N1 H1 O6 2_546 0.94(3) 1.96(3) 2.8510(19) 156(3) yes O2 H2 O1 1_655 0.86(3) 1.89(3) 2.7408(17) 169(3) yes O5 H3 O2 1_565 0.91(4) 1.86(4) 2.7338(18) 161(3) yes O6 H4 O5 1_455 0.93(3) 1.75(3) 2.6610(18) 167(3) yes loop_ _cod_related_entry_id _cod_related_entry_database _cod_related_entry_code 1 ChemSpider 21173882 2 PubChem 57408444