#------------------------------------------------------------------------------ #$Date: 2016-02-14 04:40:26 +0000 (Sun, 14 Feb 2016) $ #$Revision: 176432 $ #$URL: svn://www.crystallography.net/cod/cif/2/20/68/2206839.cif $ #------------------------------------------------------------------------------ # # This file is available in the Crystallography Open Database (COD), # http://www.crystallography.net/. The original data for this entry # were provided by IUCr Journals, http://journals.iucr.org/. # # The file may be used within the scientific community so long as # proper attribution is given to the journal article from which the # data were obtained. # data_2206839 loop_ _publ_author_name 'Sonar, Vijayakumar N.' 'Parkin, Sean' 'Crooks, Peter A.' _publ_section_title (2E,4E)-8-Methyl-2,4-bis(3-thienylmethylene)-8-azabicyclo[3.2.1]octan-3-one _journal_coeditor_code AC6202 _journal_issue 10 _journal_name_full 'Acta Crystallographica Section E' _journal_page_first o3445 _journal_page_last o3446 _journal_paper_doi 10.1107/S160053680503028X _journal_volume 61 _journal_year 2005 _chemical_formula_iupac 'C18 H17 N O S2' _chemical_formula_moiety 'C18 H17 N O S2' _chemical_formula_sum 'C18 H17 N O S2' _chemical_formula_weight 327.45 _chemical_name_systematic (2E,4E)-8-Methyl-2,4-bis-thiophen-3-ylmethylene-8-azabicyclo[3.2.1]octan-3-one _space_group_IT_number 36 _symmetry_cell_setting orthorhombic _symmetry_space_group_name_Hall 'C 2c -2' _symmetry_space_group_name_H-M 'C m c 21' _atom_sites_solution_hydrogens geom _atom_sites_solution_primary direct _atom_sites_solution_secondary difmap _audit_creation_method SHELXL97 _cell_angle_alpha 90.00 _cell_angle_beta 90.00 _cell_angle_gamma 90.00 _cell_formula_units_Z 4 _cell_length_a 19.3783(4) _cell_length_b 10.5680(6) _cell_length_c 7.3257(3) _cell_measurement_reflns_used 994 _cell_measurement_temperature 90.0(2) _cell_measurement_theta_max 27.48 _cell_measurement_theta_min 1.00 _cell_volume 1500.23(11) _computing_cell_refinement 'SCALEPACK (Otwinowski & Minor, 1997)' _computing_data_collection 'COLLECT (Nonius, 1999)' _computing_data_reduction 'DENZO-SMN (Otwinowski & Minor, 1997)' _computing_molecular_graphics 'XP in SHELXTL (Sheldrick, 1995)' _computing_publication_material 'SHELXL97 and local procedures' _computing_structure_refinement 'SHELXL97 (Sheldrick, 1997)' _computing_structure_solution 'SHELXS97 (Sheldrick, 1997)' _diffrn_ambient_temperature 90.0(2) _diffrn_detector_area_resol_mean 18 _diffrn_measured_fraction_theta_full 0.997 _diffrn_measured_fraction_theta_max 0.997 _diffrn_measurement_device_type 'Nonius KappaCCD area-detector' _diffrn_measurement_method '\w scans at fixed \c = 55\%' _diffrn_radiation_monochromator graphite _diffrn_radiation_source 'fine-focus sealed tube' _diffrn_radiation_type MoK\a _diffrn_radiation_wavelength 0.71073 _diffrn_reflns_av_R_equivalents 0.0360 _diffrn_reflns_av_sigmaI/netI 0.0353 _diffrn_reflns_limit_h_max 25 _diffrn_reflns_limit_h_min -24 _diffrn_reflns_limit_k_max 13 _diffrn_reflns_limit_k_min -13 _diffrn_reflns_limit_l_max 9 _diffrn_reflns_limit_l_min -9 _diffrn_reflns_number 1668 _diffrn_reflns_theta_full 27.49 _diffrn_reflns_theta_max 27.49 _diffrn_reflns_theta_min 2.10 _diffrn_standards_decay_% 0 _diffrn_standards_interval_count 0 _exptl_absorpt_coefficient_mu 0.356 _exptl_absorpt_correction_T_max 0.9486 _exptl_absorpt_correction_T_min 0.9164 _exptl_absorpt_correction_type multi-scan _exptl_absorpt_process_details '(SCALEPACK, Version 0.95.373; Otwinowski & Minor, 1997)' _exptl_crystal_colour brown _exptl_crystal_density_diffrn 1.450 _exptl_crystal_density_method 'not measured' _exptl_crystal_description 'irregular fragment' _exptl_crystal_F_000 688 _exptl_crystal_size_max 0.25 _exptl_crystal_size_mid 0.20 _exptl_crystal_size_min 0.15 _refine_diff_density_max 0.229 _refine_diff_density_min -0.196 _refine_ls_abs_structure_details 'Flack (1983), with how many Friedel pairs' _refine_ls_abs_structure_Flack 0.47(9) _refine_ls_extinction_method none _refine_ls_goodness_of_fit_ref 1.081 _refine_ls_hydrogen_treatment constr _refine_ls_matrix_type full _refine_ls_number_parameters 144 _refine_ls_number_reflns 1668 _refine_ls_number_restraints 186 _refine_ls_restrained_S_all 1.052 _refine_ls_R_factor_all 0.0363 _refine_ls_R_factor_gt 0.0313 _refine_ls_shift/su_max 0.001 _refine_ls_shift/su_mean 0.000 _refine_ls_structure_factor_coef Fsqd _refine_ls_weighting_details 'calc w = 1/[\s^2^(Fo^2^)+(0.0376P)^2^+0.3768P] where P=(Fo^2^+2Fc^2^)/3' _refine_ls_weighting_scheme calc _refine_ls_wR_factor_gt 0.0709 _refine_ls_wR_factor_ref 0.0738 _reflns_number_gt 1551 _reflns_number_total 1668 _reflns_threshold_expression I>2\s(I) _cod_data_source_file ac6202.cif _cod_data_source_block I _cod_original_sg_symbol_Hall 'C 2c -2 ' _cod_database_code 2206839 _cod_database_fobs_code 2206839 loop_ _symmetry_equiv_pos_as_xyz 'x, y, z' '-x, -y, z+1/2' '-x, y, z' 'x, -y, z+1/2' 'x+1/2, y+1/2, z' '-x+1/2, -y+1/2, z+1/2' '-x+1/2, y+1/2, z' 'x+1/2, -y+1/2, z+1/2' loop_ _atom_site_label _atom_site_fract_x _atom_site_fract_y _atom_site_fract_z _atom_site_U_iso_or_equiv _atom_site_adp_type _atom_site_calc_flag _atom_site_refinement_flags _atom_site_occupancy _atom_site_disorder_assembly _atom_site_disorder_group _atom_site_type_symbol O1 1.0000 1.04922(15) 0.7913(3) 0.0239(4) Uani d SU 1 . . O N1 1.0000 0.67138(18) 0.8054(3) 0.0157(4) Uani d SU 1 . . N C1 1.0000 0.9364(2) 0.7552(3) 0.0165(5) Uani d SU 1 . . C C2 0.93431(8) 0.86450(14) 0.7290(3) 0.0155(3) Uani d U 1 B . C C3 0.94082(8) 0.72283(14) 0.7042(3) 0.0152(3) Uani d U 1 . . C H3 0.8972 0.6795 0.7421 0.018 Uiso calc R 1 . . H C4 0.95997(8) 0.68646(16) 0.5066(3) 0.0182(4) Uani d U 1 . . C H4A 0.9417 0.7492 0.4186 0.022 Uiso calc R 1 . . H H4B 0.9417 0.6018 0.4751 0.022 Uiso calc R 1 . . H C5 1.0000 0.6941(2) 1.0032(3) 0.0201(5) Uani d SU 1 . . C H5A 0.9933 0.7846 1.0268 0.030 Uiso calc PR 0.50 . . H H5B 1.0442 0.6669 1.0549 0.030 Uiso calc PR 0.50 . . H H5C 0.9625 0.6460 1.0599 0.030 Uiso calc PR 0.50 . . H C6 0.87556(8) 0.93268(15) 0.7284(2) 0.0160(3) Uani d U 1 . . C H6 0.8813 1.0203 0.7532 0.019 Uiso calc R 1 A 1 H C7 0.80459(7) 0.89298(15) 0.6955(3) 0.0144(3) Uani d PDU 0.604(2) B 1 C C8 0.7817(6) 0.7892(12) 0.607(3) 0.0135(13) Uani d PDU 0.604(2) B 1 C H8 0.8119 0.7276 0.5566 0.016 Uiso calc PR 0.604(2) B 1 H S1 0.69352(6) 0.77756(15) 0.5917(2) 0.0162(3) Uani d PDU 0.604(2) B 1 S C9 0.6851(4) 0.9185(10) 0.7108(17) 0.0176(16) Uani d PDU 0.604(2) B 1 C H9 0.6420 0.9539 0.7448 0.021 Uiso calc PR 0.604(2) B 1 H C10 0.7459(4) 0.9719(11) 0.7496(19) 0.0136(12) Uani d PDU 0.604(2) B 1 C H10 0.7505 1.0523 0.8062 0.016 Uiso calc PR 0.604(2) B 1 H C7' 0.80459(7) 0.89298(15) 0.6955(3) 0.0144(3) Uani d PDU 0.396(2) B 2 C C8' 0.7535(6) 0.9653(16) 0.754(3) 0.0143(18) Uani d PDU 0.396(2) B 2 C H8' 0.7607 1.0396 0.8246 0.017 Uiso calc PR 0.396(2) B 2 H S1' 0.67364(15) 0.9136(4) 0.6918(6) 0.0170(5) Uani d PDU 0.396(2) B 2 S C9' 0.7115(4) 0.7811(11) 0.593(2) 0.0203(18) Uani d PDU 0.396(2) B 2 C H9' 0.6852 0.7156 0.5374 0.024 Uiso calc PR 0.396(2) B 2 H C10' 0.7801(9) 0.7786(19) 0.600(4) 0.0135(18) Uani d PDU 0.396(2) B 2 C H10' 0.8087 0.7136 0.5522 0.016 Uiso calc PR 0.396(2) B 2 H loop_ _atom_site_aniso_label _atom_site_aniso_U_11 _atom_site_aniso_U_22 _atom_site_aniso_U_33 _atom_site_aniso_U_12 _atom_site_aniso_U_13 _atom_site_aniso_U_23 O1 0.0190(8) 0.0157(8) 0.0368(10) 0.000 0.000 -0.0037(7) N1 0.0137(8) 0.0159(9) 0.0176(10) 0.000 0.000 0.0012(8) C1 0.0157(10) 0.0143(9) 0.0195(12) 0.000 0.000 -0.0001(9) C2 0.0155(7) 0.0157(7) 0.0152(9) -0.0010(6) 0.0005(6) 0.0005(6) C3 0.0126(7) 0.0141(7) 0.0188(9) -0.0009(5) -0.0010(7) 0.0001(7) C4 0.0211(9) 0.0151(7) 0.0183(9) -0.0001(6) -0.0028(7) -0.0012(7) C5 0.0194(11) 0.0224(11) 0.0185(12) 0.000 0.000 0.0005(10) C6 0.0175(7) 0.0141(7) 0.0165(9) -0.0011(6) 0.0004(6) 0.0016(7) C7 0.0154(7) 0.0144(7) 0.0135(8) 0.0017(5) -0.0004(7) 0.0037(6) C8 0.0128(16) 0.014(2) 0.014(2) 0.0028(15) 0.0004(16) 0.0019(19) S1 0.0143(5) 0.0170(4) 0.0172(4) -0.0009(4) -0.0013(5) 0.0000(3) C9 0.021(2) 0.016(2) 0.016(3) 0.0041(19) 0.002(2) -0.0008(16) C10 0.0132(19) 0.0127(18) 0.015(2) 0.0085(14) -0.0019(17) -0.0005(15) C7' 0.0154(7) 0.0144(7) 0.0135(8) 0.0017(5) -0.0004(7) 0.0037(6) C8' 0.014(2) 0.015(3) 0.014(3) -0.003(2) -0.002(2) 0.002(2) S1' 0.0120(8) 0.0204(8) 0.0186(11) -0.0020(7) -0.0007(8) 0.0004(7) C9' 0.025(3) 0.018(2) 0.018(3) -0.001(2) 0.002(3) -0.0030(18) C10' 0.017(2) 0.013(3) 0.011(3) -0.0022(19) 0.000(2) -0.002(2) loop_ _atom_type_symbol _atom_type_description _atom_type_scat_dispersion_real _atom_type_scat_dispersion_imag _atom_type_scat_source C C .0033 .0016 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' H H .0000 .0000 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' N N .0061 .0033 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' O O .0106 .0060 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' S S .1246 .1234 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' loop_ _geom_angle_atom_site_label_1 _geom_angle_atom_site_label_2 _geom_angle_atom_site_label_3 _geom_angle_site_symmetry_1 _geom_angle_site_symmetry_3 _geom_angle _geom_angle_publ_flag C5 N1 C3 . 3_755 115.92(13) ? C5 N1 C3 . . 115.92(13) ? C3 N1 C3 3_755 . 102.55(18) ? O1 C1 C2 . 3_755 121.63(9) ? O1 C1 C2 . . 121.62(9) y C2 C1 C2 3_755 . 116.72(19) ? C6 C2 C1 . . 116.60(15) y C6 C2 C3 . . 126.81(14) ? C1 C2 C3 . . 116.58(14) ? N1 C3 C2 . . 111.75(15) ? N1 C3 C4 . . 101.15(13) ? C2 C3 C4 . . 112.28(14) ? N1 C3 H3 . . 110.4 ? C2 C3 H3 . . 110.4 ? C4 C3 H3 . . 110.4 ? C3 C4 C4 . 3_755 103.92(8) ? C3 C4 H4A . . 111.0 ? C4 C4 H4A 3_755 . 111.0 ? C3 C4 H4B . . 111.0 ? C4 C4 H4B 3_755 . 111.0 ? H4A C4 H4B . . 109.0 ? N1 C5 H5A . . 109.5 ? N1 C5 H5B . . 109.5 ? H5A C5 H5B . . 109.5 ? N1 C5 H5C . . 109.5 ? H5A C5 H5C . . 109.5 ? H5B C5 H5C . . 109.5 ? C2 C6 C7 . . 130.07(14) y C2 C6 H6 . . 115.0 ? C7 C6 H6 . . 115.0 ? C8 C7 C6 . . 128.6(5) y C8 C7 C10 . . 109.7(4) ? C6 C7 C10 . . 121.6(4) ? C7 C8 S1 . . 114.6(7) y C7 C8 H8 . . 122.7 ? S1 C8 H8 . . 122.7 ? C8 S1 C9 . . 90.0(4) y C10 C9 S1 . . 112.8(7) ? C10 C9 H9 . . 123.6 ? S1 C9 H9 . . 123.6 ? C9 C10 C7 . . 112.7(8) ? C9 C10 H10 . . 123.7 ? C7 C10 H10 . . 123.7 ? S1' C8' H8' . . 123.0 ? C8' S1' C9' . . 89.2(6) ? C10' C9' S1' . . 114.8(9) ? C10' C9' H9' . . 122.6 ? S1' C9' H9' . . 122.6 ? C9' C10' H10' . . 125.5 ? loop_ _geom_bond_atom_site_label_1 _geom_bond_atom_site_label_2 _geom_bond_site_symmetry_2 _geom_bond_distance _geom_bond_publ_flag O1 C1 . 1.221(3) y N1 C5 . 1.469(3) y N1 C3 3_755 1.470(2) ? N1 C3 . 1.470(2) y C1 C2 3_755 1.4951(19) ? C1 C2 . 1.4952(19) y C2 C6 . 1.347(2) y C2 C3 . 1.513(2) y C3 C4 . 1.543(3) y C3 H3 . 1.0000 ? C4 C4 3_755 1.552(3) ? C4 H4A . 0.9900 ? C4 H4B . 0.9900 ? C5 H5A . 0.9800 ? C5 H5B . 0.9800 ? C5 H5C . 0.9800 ? C6 C7 . 1.458(2) y C6 H6 . 0.9500 ? C7 C8 . 1.350(10) ? C7 C10 . 1.465(8) ? C8 S1 . 1.716(11) y C8 H8 . 0.9500 ? S1 C9 . 1.733(9) y C9 C10 . 1.337(12) ? C9 H9 . 0.9500 ? C10 H10 . 0.9500 ? C8' S1' . 1.704(14) ? C8' H8' . 0.9500 ? S1' C9' . 1.740(10) ? C9' C10' . 1.331(18) ? C9' H9' . 0.9500 ? C10' H10' . 0.9500 ? loop_ _geom_torsion_atom_site_label_1 _geom_torsion_atom_site_label_2 _geom_torsion_atom_site_label_3 _geom_torsion_atom_site_label_4 _geom_torsion_site_symmetry_1 _geom_torsion_site_symmetry_4 _geom_torsion _geom_torsion_publ_flag O1 C1 C2 C6 . . 6.6(3) y C2 C1 C2 C6 3_755 . -171.36(13) ? O1 C1 C2 C3 . . -173.9(2) y C2 C1 C2 C3 3_755 . 8.1(3) ? C5 N1 C3 C2 . . 58.0(2) ? C3 N1 C3 C2 3_755 . -69.3(2) ? C5 N1 C3 C4 . . 177.69(15) ? C3 N1 C3 C4 3_755 . 50.38(18) ? C6 C2 C3 N1 . . -148.89(17) ? C1 C2 C3 N1 . . 31.7(2) ? C6 C2 C3 C4 . . 98.2(2) ? C1 C2 C3 C4 . . -81.18(19) ? N1 C3 C4 C4 . 3_755 -29.76(11) ? C2 C3 C4 C4 . 3_755 89.51(11) ? C1 C2 C6 C7 . . 175.88(18) ? C3 C2 C6 C7 . . -3.5(3) ? C2 C6 C7 C8 . . -21.6(12) y C2 C6 C7 C10 . . 162.7(7) y C6 C7 C8 S1 . . -178.5(5) ? C10 C7 C8 S1 . . -2.3(17) ? C7 C8 S1 C9 . . -0.2(14) ? C8 S1 C9 C10 . . 2.9(13) ? S1 C9 C10 C7 . . -4.8(15) ? C8 C7 C10 C9 . . 4.6(17) ? C6 C7 C10 C9 . . -178.9(9) ? C8' S1' C9' C10' . . -2(2) ?