#------------------------------------------------------------------------------ #$Date: 2010-01-30 13:59:17 +0000 (Sat, 30 Jan 2010) $ #$Revision: 966 $ #$URL: svn://www.crystallography.net/cod/cif/2/2214252.cif $ #------------------------------------------------------------------------------ # # This file is available in the Crystallography Open Database (COD), # http://www.crystallography.net/. The original data for this entry # were provided by IUCr Journals, http://journals.iucr.org/. # # The file may be used within the scientific community so long as # proper attribution is given to the journal article from which the # data were obtained. # data_2214252 loop_ _publ_author_name 'Xu, Jia-Ying' 'Wu, Zhen-Yi' 'Wu, Wen-Yuan' 'Tian, Wen-Wen' 'Wang, Jin-Tang' _publ_section_title ; Methyl 3-carboxy-7-(tert-butoxycarbonyl)-4,7-diazaheptanoate ; _journal_coeditor_code HK2260 _journal_issue 7 _journal_name_full 'Acta Crystallographica, Section E' _journal_page_first o3079 _journal_page_last o3079 _journal_volume 63 _journal_year 2007 _chemical_formula_iupac 'C12 H22 N2 O6' _chemical_formula_moiety 'C12 H22 N2 O6' _chemical_formula_sum 'C12 H22 N2 O6' _chemical_formula_weight 290.32 _chemical_melting_point 454 _chemical_name_systematic ; Methyl 3-carboxy-7-(tert-butoxycarbonyl)-4,7-diazaheptanoate ; _symmetry_cell_setting orthorhombic _symmetry_space_group_name_Hall 'P 2c -2ac' _symmetry_space_group_name_H-M 'P c a 21' _atom_sites_solution_hydrogens geom _atom_sites_solution_primary direct _atom_sites_solution_secondary difmap _audit_creation_method SHELXL97 _cell_angle_alpha 90 _cell_angle_beta 90 _cell_angle_gamma 90 _cell_formula_units_Z 4 _cell_length_a 10.824(2) _cell_length_b 15.204(3) _cell_length_c 8.9300(18) _cell_measurement_reflns_used 25 _cell_measurement_temperature 298(2) _cell_measurement_theta_max 12 _cell_measurement_theta_min 9 _cell_volume 1469.6(5) _computing_cell_refinement 'CAD-4 Software' _computing_data_collection 'CAD-4 Software (Enraf--Nonius, 1989)' _computing_data_reduction 'XCAD4 (Harms & Wocadlo, 1995)' _computing_molecular_graphics 'SHELXTL (Bruker, 2000)' _computing_publication_material SHELXTL _computing_structure_refinement 'SHELXL97 (Sheldrick, 1997)' _computing_structure_solution 'SHELXS97 (Sheldrick, 1997)' _diffrn_ambient_temperature 298(2) _diffrn_measured_fraction_theta_full 0.999 _diffrn_measured_fraction_theta_max 0.999 _diffrn_measurement_device_type 'Enraf--Nonius CAD-4' _diffrn_measurement_method \w/2\q _diffrn_radiation_monochromator graphite _diffrn_radiation_source 'fine-focus sealed tube' _diffrn_radiation_type MoK\a _diffrn_radiation_wavelength 0.71073 _diffrn_reflns_av_R_equivalents 0.0417 _diffrn_reflns_av_sigmaI/netI 0.0553 _diffrn_reflns_limit_h_max 13 _diffrn_reflns_limit_h_min 0 _diffrn_reflns_limit_k_max 18 _diffrn_reflns_limit_k_min 0 _diffrn_reflns_limit_l_max 10 _diffrn_reflns_limit_l_min 0 _diffrn_reflns_number 1921 _diffrn_reflns_theta_full 25.96 _diffrn_reflns_theta_max 25.96 _diffrn_reflns_theta_min 1.34 _diffrn_standards_decay_% 0 _diffrn_standards_interval_count 200 _diffrn_standards_number 3 _exptl_absorpt_coefficient_mu 0.105 _exptl_absorpt_correction_T_max 0.9896 _exptl_absorpt_correction_T_min 0.9542 _exptl_absorpt_correction_type psi-scan _exptl_absorpt_process_details '(North et al., 1968)' _exptl_crystal_colour colourless _exptl_crystal_density_diffrn 1.312 _exptl_crystal_density_method 'not measured' _exptl_crystal_description block _exptl_crystal_F_000 624 _exptl_crystal_size_max 0.40 _exptl_crystal_size_mid 0.30 _exptl_crystal_size_min 0.10 _refine_diff_density_max 0.228 _refine_diff_density_min -0.130 _refine_ls_extinction_method none _refine_ls_goodness_of_fit_ref 0.898 _refine_ls_hydrogen_treatment constr _refine_ls_matrix_type full _refine_ls_number_parameters 182 _refine_ls_number_reflns 1540 _refine_ls_number_restraints 0 _refine_ls_restrained_S_all 0.898 _refine_ls_R_factor_all 0.0981 _refine_ls_R_factor_gt 0.0574 _refine_ls_shift/su_max 0.000 _refine_ls_shift/su_mean 0.000 _refine_ls_structure_factor_coef Fsqd _refine_ls_weighting_details 'calc w = 1/[\s^2^(Fo^2^)+(0.059P)^2^+3.5659P] where P=(Fo^2^+2Fc^2^)/3' _refine_ls_weighting_scheme calc _refine_ls_wR_factor_gt 0.1029 _refine_ls_wR_factor_ref 0.1293 _reflns_number_gt 984 _reflns_number_total 1540 _reflns_threshold_expression I>2\s(I) _[local]_cod_data_source_file hk2260.cif loop_ _symmetry_equiv_pos_as_xyz 'x, y, z' '-x, -y, z+1/2' 'x+1/2, -y, z' '-x+1/2, y, z+1/2' loop_ _atom_type_symbol _atom_type_description _atom_type_scat_dispersion_real _atom_type_scat_dispersion_imag _atom_type_scat_source C C 0.0033 0.0016 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' H H 0.0000 0.0000 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' N N 0.0061 0.0033 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' O O 0.0106 0.0060 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' loop_ _atom_site_type_symbol _atom_site_label _atom_site_fract_x _atom_site_fract_y _atom_site_fract_z _atom_site_U_iso_or_equiv _atom_site_adp_type _atom_site_calc_flag _atom_site_refinement_flags _atom_site_occupancy O O1 0.9191(4) 0.8093(3) 0.6834(6) 0.0502(12) Uani d . 1 O O2 0.9209(5) 0.8738(3) 0.4545(6) 0.0675(15) Uani d . 1 O O3 1.1376(4) 0.4304(3) 0.1506(6) 0.0587(15) Uani d . 1 H H3 1.2097 0.4253 0.1777 0.088 Uiso calc R 1 O O4 1.1218(3) 0.5130(3) 0.3553(5) 0.0538(12) Uani d . 1 O O5 0.8910(4) 0.3791(3) 0.4610(6) 0.0600(13) Uani d . 1 O O6 0.7747(4) 0.2899(3) 0.3195(6) 0.0562(13) Uani d . 1 N N1 0.8734(5) 0.7303(4) 0.4871(7) 0.0542(15) Uani d . 1 H H1 0.8748 0.6869 0.5487 0.065 Uiso calc R 1 N N2 0.8842(4) 0.5550(3) 0.3022(6) 0.0385(13) Uani d . 1 H H2 0.8391 0.5417 0.3782 0.046 Uiso calc R 1 C C1 0.8483(4) 0.9585(4) 0.7424(5) 0.072(3) Uani d . 1 H H1B 0.8520 0.9787 0.6407 0.108 Uiso calc R 1 H H1C 0.8605 1.0072 0.8091 0.108 Uiso calc R 1 H H1A 0.7690 0.9325 0.7610 0.108 Uiso calc R 1 C C2 0.9464(4) 0.8585(4) 0.9272(5) 0.070(3) Uani d . 1 H H2B 1.0113 0.8162 0.9403 0.105 Uiso calc R 1 H H2C 0.8682 0.8314 0.9484 0.105 Uiso calc R 1 H H2A 0.9591 0.9070 0.9944 0.105 Uiso calc R 1 C C3 1.0736(4) 0.9238(4) 0.7211(4) 0.070(2) Uani d . 1 H H3A 1.0700 0.9451 0.6200 0.105 Uiso calc R 1 H H3B 1.1318 0.8763 0.7272 0.105 Uiso calc R 1 H H3C 1.0991 0.9706 0.7864 0.105 Uiso calc R 1 C C4 0.9472(4) 0.8915(4) 0.7681(5) 0.055(2) Uani d . 1 C C5 0.9062(4) 0.8111(4) 0.5360(5) 0.0466(17) Uani d . 1 C C6 0.8359(4) 0.7149(4) 0.3337(4) 0.065(2) Uani d . 1 H H6A 0.8419 0.7698 0.2786 0.078 Uiso calc R 1 H H6B 0.7499 0.6969 0.3328 0.078 Uiso calc R 1 C C7 0.9117(4) 0.6461(4) 0.2543(4) 0.0552(19) Uani d . 1 H H7A 0.8972 0.6509 0.1474 0.066 Uiso calc R 1 H H7B 0.9986 0.6579 0.2720 0.066 Uiso calc R 1 C C8 0.9439(4) 0.4897(4) 0.2033(4) 0.0359(14) Uani d . 1 H H8 0.9422 0.5149 0.1023 0.043 Uiso calc R 1 C C9 1.0804(4) 0.4764(4) 0.2425(5) 0.0365(14) Uani d . 1 C C10 0.8706(4) 0.4040(4) 0.1954(4) 0.0362(14) Uani d . 1 H H10A 0.7907 0.4162 0.1507 0.043 Uiso d R 1 H H10B 0.9209 0.3647 0.1354 0.043 Uiso d R 1 C C11 0.8504(4) 0.3591(4) 0.3417(4) 0.0420(15) Uani d . 1 C C12 0.7384(4) 0.2387(4) 0.4468(5) 0.070(2) Uani d . 1 H H12A 0.8051 0.2366 0.5175 0.105 Uiso calc R 1 H H12B 0.7182 0.1801 0.4152 0.105 Uiso calc R 1 H H12C 0.6674 0.2652 0.4931 0.105 Uiso calc R 1 loop_ _atom_site_aniso_label _atom_site_aniso_U_11 _atom_site_aniso_U_22 _atom_site_aniso_U_33 _atom_site_aniso_U_12 _atom_site_aniso_U_13 _atom_site_aniso_U_23 O1 0.046(3) 0.045(2) 0.059(3) -0.009(2) -0.003(3) -0.002(2) O2 0.086(4) 0.050(3) 0.067(4) -0.005(3) 0.000(3) 0.013(3) O3 0.025(2) 0.052(3) 0.099(4) 0.002(2) 0.016(3) -0.012(3) O4 0.0221(18) 0.092(4) 0.047(3) -0.010(2) -0.008(2) 0.009(3) O5 0.049(3) 0.076(3) 0.055(3) -0.013(2) -0.007(3) -0.005(3) O6 0.049(3) 0.058(3) 0.062(3) -0.015(2) 0.010(3) -0.010(3) N1 0.061(4) 0.048(3) 0.053(4) 0.008(3) -0.009(3) -0.006(3) N2 0.020(2) 0.050(3) 0.045(3) 0.001(2) -0.001(2) 0.002(3) C1 0.051(5) 0.067(5) 0.102(9) 0.024(4) -0.010(6) -0.022(6) C2 0.049(4) 0.087(7) 0.074(6) -0.011(4) 0.004(4) -0.028(5) C3 0.045(4) 0.061(4) 0.104(7) -0.006(3) -0.008(5) -0.008(5) C4 0.034(3) 0.047(4) 0.082(6) 0.002(3) -0.007(4) -0.018(4) C5 0.027(3) 0.061(5) 0.052(4) 0.005(3) 0.003(3) 0.008(4) C6 0.071(5) 0.067(5) 0.059(5) 0.025(4) -0.011(5) -0.002(5) C7 0.076(5) 0.049(4) 0.041(4) 0.011(4) -0.002(4) 0.006(3) C8 0.018(2) 0.045(3) 0.044(4) 0.001(2) 0.001(3) 0.000(3) C9 0.018(2) 0.047(3) 0.044(4) 0.005(3) -0.001(3) 0.002(3) C10 0.021(3) 0.052(3) 0.036(3) -0.001(3) -0.001(3) -0.008(3) C11 0.020(3) 0.052(4) 0.054(4) 0.003(3) 0.002(3) -0.016(4) C12 0.058(4) 0.070(4) 0.083(6) -0.004(4) 0.029(5) -0.002(5) loop_ _geom_bond_atom_site_label_1 _geom_bond_atom_site_label_2 _geom_bond_distance O1 C5 1.324(8) O1 C4 1.492(8) O2 C5 1.211(8) O3 C9 1.244(7) O3 H3 0.8200 O4 C9 1.235(7) O5 C11 1.192(8) O6 C11 1.348(7) O6 C12 1.433(8) N1 C5 1.351(8) N1 C6 1.448(10) N1 H1 0.8600 N2 C8 1.477(7) N2 C7 1.479(8) N2 H2 0.8600 C1 C4 1.495(9) C1 H1B 0.9600 C1 H1C 0.9600 C1 H1A 0.9600 C2 C4 1.507(11) C2 H2B 0.9600 C2 H2C 0.9600 C2 H2A 0.9600 C3 C4 1.513(9) C3 H3A 0.9600 C3 H3B 0.9600 C3 H3C 0.9600 C6 C7 1.508(9) C6 H6A 0.9700 C6 H6B 0.9700 C7 H7A 0.9700 C7 H7B 0.9700 C8 C9 1.531(7) C8 C10 1.528(7) C8 H8 0.9800 C10 C11 1.491(9) C10 H10A 0.9700 C10 H10B 0.9701 C12 H12A 0.9600 C12 H12B 0.9600 C12 H12C 0.9600 loop_ _geom_angle_atom_site_label_1 _geom_angle_atom_site_label_2 _geom_angle_atom_site_label_3 _geom_angle C5 O1 C4 120.5(6) C9 O3 H3 109.5 C11 O6 C12 118.3(6) C5 N1 C6 121.8(6) C5 N1 H1 119.1 C6 N1 H1 119.1 C8 N2 C7 111.6(5) C8 N2 H2 124.2 C7 N2 H2 124.2 C4 C1 H1B 109.5 C4 C1 H1C 109.5 H1B C1 H1C 109.5 C4 C1 H1A 109.5 H1B C1 H1A 109.5 H1C C1 H1A 109.5 C4 C2 H2B 109.5 C4 C2 H2C 109.5 H2B C2 H2C 109.5 C4 C2 H2A 109.5 H2B C2 H2A 109.5 H2C C2 H2A 109.5 C4 C3 H3A 109.5 C4 C3 H3B 109.5 H3A C3 H3B 109.5 C4 C3 H3C 109.5 H3A C3 H3C 109.5 H3B C3 H3C 109.5 O1 C4 C1 110.3(6) O1 C4 C2 101.5(6) C1 C4 C2 111.5(7) O1 C4 C3 108.4(6) C1 C4 C3 112.5(6) C2 C4 C3 112.0(6) O2 C5 O1 126.9(7) O2 C5 N1 123.8(7) O1 C5 N1 109.3(6) N1 C6 C7 113.8(6) N1 C6 H6A 108.8 C7 C6 H6A 108.8 N1 C6 H6B 108.8 C7 C6 H6B 108.8 H6A C6 H6B 107.7 N2 C7 C6 113.8(6) N2 C7 H7A 108.8 C6 C7 H7A 108.8 N2 C7 H7B 108.8 C6 C7 H7B 108.8 H7A C7 H7B 107.7 N2 C8 C9 112.0(5) N2 C8 C10 111.9(4) C9 C8 C10 113.5(5) N2 C8 H8 106.3 C9 C8 H8 106.3 C10 C8 H8 106.3 O4 C9 O3 127.6(5) O4 C9 C8 118.5(5) O3 C9 C8 113.9(6) C11 C10 C8 115.2(5) C11 C10 H10A 108.5 C8 C10 H10A 108.6 C11 C10 H10B 106.5 C8 C10 H10B 105.1 H10A C10 H10B 113.0 O5 C11 O6 123.7(7) O5 C11 C10 127.8(5) O6 C11 C10 108.5(6) O6 C12 H12A 109.5 O6 C12 H12B 109.5 H12A C12 H12B 109.5 O6 C12 H12C 109.5 H12A C12 H12C 109.5 H12B C12 H12C 109.5 loop_ _geom_torsion_atom_site_label_1 _geom_torsion_atom_site_label_2 _geom_torsion_atom_site_label_3 _geom_torsion_atom_site_label_4 _geom_torsion C5 O1 C4 C1 58.8(9) C5 O1 C4 C2 177.1(6) C5 O1 C4 C3 -64.9(7) C4 O1 C5 O2 4.1(10) C4 O1 C5 N1 -176.0(5) C6 N1 C5 O2 -8.8(10) C6 N1 C5 O1 171.2(6) C5 N1 C6 C7 123.3(7) C8 N2 C7 C6 169.8(5) N1 C6 C7 N2 74.1(8) C7 N2 C8 C9 80.5(6) C7 N2 C8 C10 -150.7(5) N2 C8 C9 O4 6.5(8) C10 C8 C9 O4 -121.5(6) N2 C8 C9 O3 -171.6(5) C10 C8 C9 O3 60.5(7) N2 C8 C10 C11 -58.4(6) C9 C8 C10 C11 69.6(6) C12 O6 C11 O5 1.6(8) C12 O6 C11 C10 -177.6(5) C8 C10 C11 O5 -5.2(8) C8 C10 C11 O6 173.9(4) loop_ _geom_hbond_atom_site_label_D _geom_hbond_atom_site_label_H _geom_hbond_atom_site_label_A _geom_hbond_site_symmetry_A _geom_hbond_distance_DH _geom_hbond_distance_HA _geom_hbond_distance_DA _geom_hbond_angle_DHA O3 H3 N2 3_565 0.82 2.21 3.001(6) 161 N1 H1 O3 2_765 0.86 2.01 2.849(8) 166 N2 H2 O3 2_765 0.86 2.48 3.128(8) 132 N2 H2 O4 3_465 0.86 2.50 3.060(6) 123 _cod_database_code 2214252