#------------------------------------------------------------------------------ #$Date: 2016-02-21 00:03:34 +0000 (Sun, 21 Feb 2016) $ #$Revision: 176798 $ #$URL: svn://www.crystallography.net/cod/cif/2/23/90/2239053.cif $ #------------------------------------------------------------------------------ # # This file is available in the Crystallography Open Database (COD), # http://www.crystallography.net/ # # All data on this site have been placed in the public domain by the # contributors. # data_2239053 loop_ _publ_author_name 'Govindan, E.' 'Yuvaraj, PanneerSelvam' 'Reddy, Boreddy Siva Rami' 'Premalatha, K.' 'SubbiahPandi, A.' _publ_section_title ; (4S)-5'-Chloro-3,7,7-trimethyl-5,6,7,8-tetrahydro-4H-spiro[1,2-oxazolo[5,4-b]quinoline-4,3'-indole]-2',5-dione ; _journal_coeditor_code CV5438 _journal_issue 2 _journal_name_full 'Acta Crystallographica Section E' _journal_page_first o173 _journal_paper_doi 10.1107/S1600536814000191 _journal_volume 70 _journal_year 2014 _chemical_formula_iupac 'C20 H18 Cl N3 O3' _chemical_formula_moiety 'C20 H18 Cl N3 O3' _chemical_formula_sum 'C20 H18 Cl N3 O3' _chemical_formula_weight 383.82 _chemical_name_systematic (4S)-5'-Chloro-3,7,7-trimethyl-5,6,7,8-tetrahydro-4H-spiro[1,2-oxazolo[5,4-b]quinoline-4,3'-indole]-2',5-dione _space_group_IT_number 61 _symmetry_cell_setting orthorhombic _symmetry_space_group_name_Hall '-P 2ac 2ab' _symmetry_space_group_name_H-M 'P b c a' _atom_sites_solution_hydrogens geom _atom_sites_solution_primary direct _atom_sites_solution_secondary difmap _audit_creation_method SHELXL-97 _cell_angle_alpha 90.00 _cell_angle_beta 90.00 _cell_angle_gamma 90.00 _cell_formula_units_Z 8 _cell_length_a 17.9320(7) _cell_length_b 11.1120(4) _cell_length_c 18.5968(7) _cell_measurement_reflns_used 2643 _cell_measurement_temperature 293(2) _cell_measurement_theta_max 28.34 _cell_measurement_theta_min 2.19 _cell_volume 3705.6(2) _computing_cell_refinement 'SAINT (Bruker, 2008)' _computing_data_collection 'APEX2 (Bruker, 2008)' _computing_data_reduction 'SAINT (Bruker, 2008)' _computing_molecular_graphics 'ORTEP-3 for Windows (Farrugia, 2012)' _computing_publication_material 'SHELXL97 (Sheldrick, 2008) and PLATON (Spek, 2009)' _computing_structure_refinement 'SHELXL97 (Sheldrick, 2008)' _computing_structure_solution 'SHELXS97 (Sheldrick, 2008)' _diffrn_ambient_temperature 293(2) _diffrn_measured_fraction_theta_full 0.992 _diffrn_measured_fraction_theta_max 0.992 _diffrn_measurement_device_type 'Bruker SMART APEXII CCD' _diffrn_measurement_method '\w and \f scans' _diffrn_radiation_monochromator graphite _diffrn_radiation_source 'fine-focus sealed tube' _diffrn_radiation_type MoK\a _diffrn_radiation_wavelength 0.71073 _diffrn_reflns_av_R_equivalents 0.0316 _diffrn_reflns_av_sigmaI/netI 0.0384 _diffrn_reflns_limit_h_max 23 _diffrn_reflns_limit_h_min -22 _diffrn_reflns_limit_k_max 12 _diffrn_reflns_limit_k_min -14 _diffrn_reflns_limit_l_max 24 _diffrn_reflns_limit_l_min -24 _diffrn_reflns_number 17841 _diffrn_reflns_theta_full 28.34 _diffrn_reflns_theta_max 28.34 _diffrn_reflns_theta_min 2.19 _exptl_absorpt_coefficient_mu 0.232 _exptl_absorpt_correction_T_max 0.959 _exptl_absorpt_correction_T_min 0.952 _exptl_absorpt_correction_type multi-scan _exptl_absorpt_process_details '(SADABS; Bruker, 2008)' _exptl_crystal_colour White _exptl_crystal_density_diffrn 1.376 _exptl_crystal_density_method 'not measured' _exptl_crystal_description Block _exptl_crystal_F_000 1600 _exptl_crystal_size_max 0.21 _exptl_crystal_size_mid 0.19 _exptl_crystal_size_min 0.18 _refine_diff_density_max 0.285 _refine_diff_density_min -0.359 _refine_ls_extinction_method none _refine_ls_goodness_of_fit_ref 1.011 _refine_ls_hydrogen_treatment constr _refine_ls_matrix_type full _refine_ls_number_parameters 247 _refine_ls_number_reflns 4590 _refine_ls_number_restraints 0 _refine_ls_restrained_S_all 1.011 _refine_ls_R_factor_all 0.0970 _refine_ls_R_factor_gt 0.0437 _refine_ls_shift/su_max 0.000 _refine_ls_shift/su_mean 0.000 _refine_ls_structure_factor_coef Fsqd _refine_ls_weighting_details 'calc w=1/[\s^2^(Fo^2^)+(0.0522P)^2^+1.5319P] where P=(Fo^2^+2Fc^2^)/3' _refine_ls_weighting_scheme calc _refine_ls_wR_factor_gt 0.1024 _refine_ls_wR_factor_ref 0.1335 _reflns_number_gt 2643 _reflns_number_total 4590 _reflns_threshold_expression I>2sigma(I) _iucr_refine_instructions_details ; TITL aspyr15 in P b c a CELL 0.71073 17.9320 11.1120 18.5968 90.000 90.000 90.000 ZERR 8.00 0.0007 0.0004 0.0007 0.000 0.000 0.000 LATT 1 SYMM 1/2 - X, - Y, 1/2 + Z SYMM 1/2 + X, 1/2 - Y, - Z SYMM - X, 1/2 + Y, 1/2 - Z SFAC C H N O CL UNIT 160 144 24 24 8 MERG 2 FMAP 2 PLAN 25 EQIV $1 -x+1, -y+1, -z+1 HTAB N1, O3_$1 EQIV $2 -x+1, -y, -z+1 HTAB N3, O1_$2 ACTA BOND $H CONF L.S. 10 WGHT 0.052200 1.531900 FVAR 0.09838 C3 1 0.720854 0.440400 0.617848 11.00000 0.04597 0.07663 = 0.06379 -0.03388 0.01580 -0.01669 C4 1 0.707655 0.541682 0.577531 11.00000 0.06813 0.05886 = 0.08852 -0.03274 0.03368 -0.03301 AFIX 43 H4 2 0.734139 0.611718 0.587403 11.00000 -1.20000 AFIX 0 C5 1 0.656053 0.541610 0.522847 11.00000 0.07360 0.03537 = 0.07441 -0.01304 0.03106 -0.01751 AFIX 43 H5 2 0.647046 0.610373 0.495694 11.00000 -1.20000 AFIX 0 C6 1 0.618328 0.436451 0.509780 11.00000 0.05476 0.02964 = 0.04778 -0.00684 0.01844 -0.00744 C7 1 0.533053 0.302271 0.466742 11.00000 0.05607 0.02273 = 0.03269 0.00166 0.00954 0.00335 C8 1 0.581053 0.233602 0.522974 11.00000 0.04530 0.02436 = 0.03207 -0.00188 0.00283 -0.00004 C1 1 0.631639 0.333348 0.549838 11.00000 0.04745 0.03256 = 0.04130 -0.00942 0.01024 -0.00370 C2 1 0.682612 0.333577 0.604842 11.00000 0.04359 0.05064 = 0.05056 -0.01841 0.00734 -0.00147 AFIX 43 H2 2 0.691275 0.265092 0.632348 11.00000 -1.20000 AFIX 0 C11 1 0.707090 0.229393 0.384844 11.00000 0.07136 0.05776 = 0.06455 -0.00219 0.02262 -0.00678 AFIX 137 H11A 2 0.739675 0.197193 0.348685 11.00000 -1.50000 H11B 2 0.734764 0.282108 0.415837 11.00000 -1.50000 H11C 2 0.667520 0.273566 0.362210 11.00000 -1.50000 AFIX 0 C10 1 0.675031 0.129148 0.427922 11.00000 0.04366 0.04544 = 0.03983 -0.00710 0.00029 0.00028 N2 3 0.695041 0.018001 0.413109 11.00000 0.05584 0.04946 = 0.04836 -0.00933 0.00427 0.00467 C12 1 0.614640 0.017740 0.504158 11.00000 0.04567 0.02936 = 0.03571 -0.00561 -0.00506 0.00461 C9 1 0.622997 0.133891 0.485353 11.00000 0.04246 0.02970 = 0.03355 -0.00380 -0.00183 0.00069 C14 1 0.533388 0.176529 0.581956 11.00000 0.04506 0.02500 = 0.02849 0.00047 -0.00092 -0.00022 C13 1 0.533199 0.056682 0.598239 11.00000 0.04452 0.02782 = 0.03028 -0.00090 -0.00610 -0.00117 N3 3 0.572357 -0.025622 0.558691 11.00000 0.06130 0.02215 = 0.03953 0.00125 -0.00191 0.00385 AFIX 43 H3 2 0.570239 -0.101353 0.568002 11.00000 -1.20000 AFIX 0 C18 1 0.490514 0.005726 0.660150 11.00000 0.05778 0.03019 = 0.03779 0.00734 -0.00376 -0.00503 AFIX 23 H18A 2 0.519055 -0.059683 0.681023 11.00000 -1.20000 H18B 2 0.444049 -0.027615 0.642364 11.00000 -1.20000 AFIX 0 C17 1 0.472985 0.097379 0.718915 11.00000 0.05688 0.03954 = 0.03266 0.00492 0.00334 -0.00244 C16 1 0.438748 0.207207 0.681958 11.00000 0.05406 0.03921 = 0.04183 0.00232 0.00768 0.00177 AFIX 23 H16A 2 0.389860 0.185437 0.663814 11.00000 -1.20000 H16B 2 0.431904 0.270154 0.717488 11.00000 -1.20000 AFIX 0 C15 1 0.484205 0.256414 0.621122 11.00000 0.04740 0.02842 = 0.03370 -0.00064 -0.00135 0.00015 C20 1 0.543164 0.132658 0.759661 11.00000 0.07417 0.06513 = 0.03612 -0.00246 -0.00639 -0.00300 AFIX 137 H20A 2 0.530832 0.190732 0.795983 11.00000 -1.50000 H20B 2 0.578608 0.166922 0.726835 11.00000 -1.50000 H20C 2 0.564364 0.062595 0.781894 11.00000 -1.50000 AFIX 0 C19 1 0.416798 0.043811 0.771222 11.00000 0.07551 0.06556 = 0.05204 0.01789 0.01547 -0.00351 AFIX 137 H19A 2 0.437390 -0.027400 0.792669 11.00000 -1.50000 H19B 2 0.371885 0.023541 0.745872 11.00000 -1.50000 H19C 2 0.405672 0.101498 0.808122 11.00000 -1.50000 AFIX 0 N1 3 0.562184 0.414214 0.459386 11.00000 0.07118 0.02339 = 0.04331 0.00628 0.00981 -0.00201 AFIX 43 H1 2 0.547838 0.465352 0.427550 11.00000 -1.20000 AFIX 0 O2 4 0.655282 -0.056436 0.463643 11.00000 0.05800 0.03555 = 0.04740 -0.00856 0.00024 0.01023 O1 4 0.480470 0.261806 0.432885 11.00000 0.06297 0.03286 = 0.04177 0.00523 -0.00820 -0.00072 O3 4 0.478285 0.362267 0.603212 11.00000 0.07264 0.02649 = 0.05077 0.00400 0.01123 0.00724 CL1 5 0.784689 0.445235 0.687874 11.00000 0.06289 0.14861 = 0.09380 -0.05147 -0.00283 -0.03201 HKLF 4 REM aspyr15 in P b c a REM R1 = 0.0437 for 2643 Fo > 4sig(Fo) and 0.0970 for all 4590 data REM 247 parameters refined using 0 restraints END WGHT 0.0522 1.5322 REM Highest difference peak 0.285, deepest hole -0.359, 1-sigma level 0.045 Q1 1 0.7876 0.4768 0.6772 11.00000 0.05 0.28 Q2 1 0.8139 0.3716 0.6733 11.00000 0.05 0.22 Q3 1 0.6084 0.2807 0.5424 11.00000 0.05 0.21 Q4 1 0.5656 0.2044 0.5580 11.00000 0.05 0.20 Q5 1 0.7727 0.1993 0.3816 11.00000 0.05 0.20 Q6 1 0.6230 0.1338 0.4390 11.00000 0.05 0.20 Q7 1 0.6755 0.1438 0.4757 11.00000 0.05 0.19 Q8 1 0.6346 0.3468 0.5870 11.00000 0.05 0.18 Q9 1 0.7767 0.4379 0.6370 11.00000 0.05 0.18 Q10 1 0.6038 0.1825 0.5025 11.00000 0.05 0.18 Q11 1 0.7372 0.4307 0.7166 11.00000 0.05 0.17 Q12 1 0.5493 0.1413 0.8150 11.00000 0.05 0.16 Q13 1 0.3709 -0.0269 0.7321 11.00000 0.05 0.16 Q14 1 0.7227 0.4439 0.6619 11.00000 0.05 0.16 Q15 1 0.3678 0.0469 0.7583 11.00000 0.05 0.16 Q16 1 0.8388 0.4544 0.6381 11.00000 0.05 0.16 Q17 1 0.6950 0.2350 0.3289 11.00000 0.05 0.16 Q18 1 0.6176 0.1807 0.3938 11.00000 0.05 0.16 Q19 1 0.4610 0.1433 0.7054 11.00000 0.05 0.15 Q20 1 0.4636 0.2254 0.6497 11.00000 0.05 0.15 Q21 1 0.3979 0.2625 0.7098 11.00000 0.05 0.15 Q22 1 0.6414 -0.0523 0.5916 11.00000 0.05 0.15 Q23 1 0.4545 0.0730 0.7436 11.00000 0.05 0.15 Q24 1 0.5291 0.2194 0.6124 11.00000 0.05 0.15 Q25 1 0.5350 0.0173 0.5681 11.00000 0.05 0.15 ; _cod_data_source_file cv5438sup1.cif _cod_data_source_block I _cod_database_code 2239053 _cod_database_fobs_code 2239053 loop_ _symmetry_equiv_pos_as_xyz 'x, y, z' '-x+1/2, -y, z+1/2' 'x+1/2, -y+1/2, -z' '-x, y+1/2, -z+1/2' '-x, -y, -z' 'x-1/2, y, -z-1/2' '-x-1/2, y-1/2, z' 'x, -y-1/2, z-1/2' loop_ _atom_site_type_symbol _atom_site_label _atom_site_fract_x _atom_site_fract_y _atom_site_fract_z _atom_site_U_iso_or_equiv _atom_site_adp_type _atom_site_calc_flag _atom_site_refinement_flags _atom_site_occupancy _atom_site_symmetry_multiplicity C C3 0.72085(13) 0.4404(3) 0.61785(14) 0.0621(7) Uani d . 1 1 C C4 0.70766(15) 0.5417(3) 0.57753(16) 0.0718(8) Uani d . 1 1 H H4 0.7341 0.6117 0.5874 0.086 Uiso calc R 1 1 C C5 0.65605(15) 0.5416(2) 0.52285(14) 0.0611(7) Uani d . 1 1 H H5 0.6470 0.6104 0.4957 0.073 Uiso calc R 1 1 C C6 0.61833(12) 0.43645(18) 0.50978(11) 0.0441(5) Uani d . 1 1 C C7 0.53305(12) 0.30227(16) 0.46674(10) 0.0372(5) Uani d . 1 1 C C8 0.58105(11) 0.23360(16) 0.52297(9) 0.0339(4) Uani d . 1 1 C C1 0.63164(11) 0.33335(17) 0.54984(11) 0.0404(5) Uani d . 1 1 C C2 0.68261(11) 0.3336(2) 0.60484(12) 0.0483(5) Uani d . 1 1 H H2 0.6913 0.2651 0.6323 0.058 Uiso calc R 1 1 C C11 0.70709(15) 0.2294(2) 0.38484(14) 0.0646(7) Uani d . 1 1 H H11A 0.7397 0.1972 0.3487 0.097 Uiso calc R 1 1 H H11B 0.7348 0.2821 0.4158 0.097 Uiso calc R 1 1 H H11C 0.6675 0.2736 0.3622 0.097 Uiso calc R 1 1 C C10 0.67503(11) 0.12915(19) 0.42792(11) 0.0430(5) Uani d . 1 1 N N2 0.69504(10) 0.01800(17) 0.41311(10) 0.0512(5) Uani d . 1 1 C C12 0.61464(11) 0.01774(17) 0.50416(10) 0.0369(4) Uani d . 1 1 C C9 0.62300(11) 0.13389(16) 0.48535(10) 0.0352(4) Uani d . 1 1 C C14 0.53339(10) 0.17653(16) 0.58196(9) 0.0328(4) Uani d . 1 1 C C13 0.53320(11) 0.05668(16) 0.59824(9) 0.0342(4) Uani d . 1 1 N N3 0.57236(9) -0.02562(14) 0.55869(8) 0.0410(4) Uani d . 1 1 H H3 0.5702 -0.1014 0.5680 0.049 Uiso calc R 1 1 C C18 0.49051(12) 0.00573(18) 0.66015(10) 0.0419(5) Uani d . 1 1 H H18A 0.5191 -0.0597 0.6810 0.050 Uiso calc R 1 1 H H18B 0.4440 -0.0276 0.6424 0.050 Uiso calc R 1 1 C C17 0.47298(12) 0.09738(19) 0.71891(10) 0.0430(5) Uani d . 1 1 C C16 0.43875(12) 0.20721(19) 0.68196(11) 0.0450(5) Uani d . 1 1 H H16A 0.3899 0.1854 0.6638 0.054 Uiso calc R 1 1 H H16B 0.4319 0.2702 0.7175 0.054 Uiso calc R 1 1 C C15 0.48421(11) 0.25641(17) 0.62112(10) 0.0365(4) Uani d . 1 1 C C20 0.54316(14) 0.1327(2) 0.75966(12) 0.0585(6) Uani d . 1 1 H H20A 0.5308 0.1907 0.7960 0.088 Uiso calc R 1 1 H H20B 0.5786 0.1669 0.7268 0.088 Uiso calc R 1 1 H H20C 0.5644 0.0626 0.7819 0.088 Uiso calc R 1 1 C C19 0.41680(15) 0.0438(2) 0.77122(13) 0.0644(7) Uani d . 1 1 H H19A 0.4374 -0.0274 0.7927 0.097 Uiso calc R 1 1 H H19B 0.3719 0.0235 0.7459 0.097 Uiso calc R 1 1 H H19C 0.4057 0.1015 0.8081 0.097 Uiso calc R 1 1 N N1 0.56218(10) 0.41421(14) 0.45939(9) 0.0460(4) Uani d . 1 1 H H1 0.5478 0.4654 0.4276 0.055 Uiso calc R 1 1 O O2 0.65528(8) -0.05644(12) 0.46364(7) 0.0470(4) Uani d . 1 1 O O1 0.48047(8) 0.26181(12) 0.43288(7) 0.0459(4) Uani d . 1 1 O O3 0.47829(9) 0.36227(12) 0.60321(8) 0.0500(4) Uani d . 1 1 Cl Cl1 0.78469(4) 0.44523(9) 0.68787(4) 0.1018(3) Uani d . 1 1 loop_ _atom_site_aniso_label _atom_site_aniso_U_11 _atom_site_aniso_U_22 _atom_site_aniso_U_33 _atom_site_aniso_U_12 _atom_site_aniso_U_13 _atom_site_aniso_U_23 C3 0.0460(14) 0.0766(19) 0.0638(15) -0.0167(13) 0.0158(12) -0.0339(14) C4 0.0681(17) 0.0589(17) 0.089(2) -0.0330(14) 0.0337(16) -0.0327(15) C5 0.0736(17) 0.0354(12) 0.0744(17) -0.0175(11) 0.0311(15) -0.0130(11) C6 0.0548(13) 0.0296(11) 0.0478(11) -0.0074(9) 0.0184(10) -0.0068(9) C7 0.0561(13) 0.0227(10) 0.0327(9) 0.0033(9) 0.0095(9) 0.0017(8) C8 0.0453(11) 0.0244(9) 0.0321(9) 0.0000(8) 0.0028(8) -0.0019(7) C1 0.0475(12) 0.0326(11) 0.0413(10) -0.0037(9) 0.0102(9) -0.0094(8) C2 0.0436(12) 0.0506(13) 0.0506(12) -0.0015(10) 0.0073(10) -0.0184(10) C11 0.0714(17) 0.0578(16) 0.0646(15) -0.0068(13) 0.0226(13) -0.0022(12) C10 0.0437(12) 0.0454(13) 0.0398(11) 0.0003(10) 0.0003(9) -0.0071(9) N2 0.0558(11) 0.0495(12) 0.0484(10) 0.0047(9) 0.0043(9) -0.0093(9) C12 0.0457(12) 0.0294(10) 0.0357(10) 0.0046(9) -0.0051(9) -0.0056(8) C9 0.0425(11) 0.0297(10) 0.0335(9) 0.0007(8) -0.0018(8) -0.0038(8) C14 0.0451(11) 0.0250(9) 0.0285(9) -0.0002(8) -0.0009(8) 0.0005(7) C13 0.0445(11) 0.0278(10) 0.0303(9) -0.0012(8) -0.0061(8) -0.0009(7) N3 0.0613(11) 0.0222(8) 0.0395(9) 0.0039(7) -0.0019(8) 0.0013(7) C18 0.0578(13) 0.0302(10) 0.0378(10) -0.0050(9) -0.0038(9) 0.0073(8) C17 0.0569(13) 0.0395(11) 0.0327(10) -0.0024(10) 0.0033(9) 0.0049(8) C16 0.0541(13) 0.0392(12) 0.0418(11) 0.0018(10) 0.0077(10) 0.0023(9) C15 0.0474(11) 0.0284(10) 0.0337(9) 0.0002(8) -0.0013(9) -0.0006(8) C20 0.0742(17) 0.0651(16) 0.0361(11) -0.0030(13) -0.0064(11) -0.0025(11) C19 0.0755(17) 0.0656(16) 0.0520(13) -0.0035(13) 0.0155(13) 0.0179(12) N1 0.0712(12) 0.0234(8) 0.0433(9) -0.0020(8) 0.0098(9) 0.0063(7) O2 0.0580(9) 0.0355(8) 0.0474(8) 0.0102(7) 0.0002(7) -0.0086(6) O1 0.0630(9) 0.0329(8) 0.0418(8) -0.0007(7) -0.0082(7) 0.0052(6) O3 0.0726(10) 0.0265(7) 0.0508(9) 0.0072(7) 0.0112(8) 0.0040(6) Cl1 0.0629(5) 0.1486(8) 0.0938(6) -0.0320(5) -0.0028(4) -0.0515(5) loop_ _atom_type_symbol _atom_type_description _atom_type_scat_dispersion_real _atom_type_scat_dispersion_imag _atom_type_scat_source C C 0.0033 0.0016 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' H H 0.0000 0.0000 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' N N 0.0061 0.0033 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' O O 0.0106 0.0060 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' Cl Cl 0.1484 0.1585 'International Tables Vol C Tables 4.2.6.8 and 6.1.1.4' loop_ _geom_angle_atom_site_label_1 _geom_angle_atom_site_label_2 _geom_angle_atom_site_label_3 _geom_angle C4 C3 C2 121.3(2) C4 C3 Cl1 119.9(2) C2 C3 Cl1 118.8(2) C3 C4 C5 121.3(2) C3 C4 H4 119.4 C5 C4 H4 119.4 C6 C5 C4 117.6(2) C6 C5 H5 121.2 C4 C5 H5 121.2 C5 C6 C1 121.6(2) C5 C6 N1 128.7(2) C1 C6 N1 109.76(17) O1 C7 N1 125.72(18) O1 C7 C8 126.47(16) N1 C7 C8 107.75(17) C9 C8 C1 113.00(16) C9 C8 C14 107.84(15) C1 C8 C14 113.66(15) C9 C8 C7 108.91(14) C1 C8 C7 101.19(15) C14 C8 C7 112.14(15) C2 C1 C6 120.90(19) C2 C1 C8 130.20(19) C6 C1 C8 108.89(18) C1 C2 C3 117.3(2) C1 C2 H2 121.3 C3 C2 H2 121.3 C10 C11 H11A 109.5 C10 C11 H11B 109.5 H11A C11 H11B 109.5 C10 C11 H11C 109.5 H11A C11 H11C 109.5 H11B C11 H11C 109.5 N2 C10 C9 111.83(19) N2 C10 C11 119.01(19) C9 C10 C11 129.16(19) C10 N2 O2 105.51(16) O2 C12 C9 112.65(17) O2 C12 N3 120.60(17) C9 C12 N3 126.73(17) C12 C9 C10 103.49(17) C12 C9 C8 121.84(17) C10 C9 C8 134.67(17) C13 C14 C15 119.00(17) C13 C14 C8 124.41(16) C15 C14 C8 116.57(15) C14 C13 N3 122.11(17) C14 C13 C18 122.80(17) N3 C13 C18 115.09(16) C12 N3 C13 116.88(15) C12 N3 H3 121.6 C13 N3 H3 121.6 C13 C18 C17 113.85(16) C13 C18 H18A 108.8 C17 C18 H18A 108.8 C13 C18 H18B 108.8 C17 C18 H18B 108.8 H18A C18 H18B 107.7 C20 C17 C19 109.29(18) C20 C17 C18 111.00(18) C19 C17 C18 109.45(18) C20 C17 C16 110.52(18) C19 C17 C16 109.49(18) C18 C17 C16 107.06(16) C15 C16 C17 114.35(17) C15 C16 H16A 108.7 C17 C16 H16A 108.7 C15 C16 H16B 108.7 C17 C16 H16B 108.7 H16A C16 H16B 107.6 O3 C15 C14 120.25(17) O3 C15 C16 120.52(18) C14 C15 C16 119.19(17) C17 C20 H20A 109.5 C17 C20 H20B 109.5 H20A C20 H20B 109.5 C17 C20 H20C 109.5 H20A C20 H20C 109.5 H20B C20 H20C 109.5 C17 C19 H19A 109.5 C17 C19 H19B 109.5 H19A C19 H19B 109.5 C17 C19 H19C 109.5 H19A C19 H19C 109.5 H19B C19 H19C 109.5 C7 N1 C6 111.84(17) C7 N1 H1 124.1 C6 N1 H1 124.1 C12 O2 N2 106.51(14) loop_ _geom_bond_atom_site_label_1 _geom_bond_atom_site_label_2 _geom_bond_distance C3 C4 1.373(4) C3 C2 1.392(3) C3 Cl1 1.735(3) C4 C5 1.375(4) C4 H4 0.9300 C5 C6 1.372(3) C5 H5 0.9300 C6 C1 1.387(3) C6 N1 1.397(3) C7 O1 1.220(2) C7 N1 1.356(2) C7 C8 1.555(3) C8 C9 1.511(3) C8 C1 1.517(3) C8 C14 1.528(2) C1 C2 1.372(3) C2 H2 0.9300 C11 C10 1.488(3) C11 H11A 0.9600 C11 H11B 0.9600 C11 H11C 0.9600 C10 N2 1.315(3) C10 C9 1.419(3) N2 O2 1.441(2) C12 O2 1.333(2) C12 C9 1.346(3) C12 N3 1.355(2) C14 C13 1.366(2) C14 C15 1.448(3) C13 N3 1.368(2) C13 C18 1.494(3) N3 H3 0.8600 C18 C17 1.527(3) C18 H18A 0.9700 C18 H18B 0.9700 C17 C20 1.520(3) C17 C19 1.522(3) C17 C16 1.529(3) C16 C15 1.498(3) C16 H16A 0.9700 C16 H16B 0.9700 C15 O3 1.227(2) C20 H20A 0.9600 C20 H20B 0.9600 C20 H20C 0.9600 C19 H19A 0.9600 C19 H19B 0.9600 C19 H19C 0.9600 N1 H1 0.8600 loop_ _geom_hbond_atom_site_label_D _geom_hbond_atom_site_label_H _geom_hbond_atom_site_label_A _geom_hbond_site_symmetry_A _geom_hbond_distance_DH _geom_hbond_distance_HA _geom_hbond_distance_DA _geom_hbond_angle_DHA N1 H1 O3 5_666 0.86 2.05 2.837(2) 151 N3 H3 O1 5_656 0.86 2.00 2.795(2) 153 loop_ _geom_torsion_atom_site_label_1 _geom_torsion_atom_site_label_2 _geom_torsion_atom_site_label_3 _geom_torsion_atom_site_label_4 _geom_torsion C2 C3 C4 C5 0.1(4) Cl1 C3 C4 C5 -178.35(18) C3 C4 C5 C6 -0.2(3) C4 C5 C6 C1 -0.3(3) C4 C5 C6 N1 177.8(2) O1 C7 C8 C9 65.4(2) N1 C7 C8 C9 -111.86(17) O1 C7 C8 C1 -175.38(18) N1 C7 C8 C1 7.40(18) O1 C7 C8 C14 -53.9(2) N1 C7 C8 C14 128.87(16) C5 C6 C1 C2 0.9(3) N1 C6 C1 C2 -177.55(17) C5 C6 C1 C8 179.47(18) N1 C6 C1 C8 1.1(2) C9 C8 C1 C2 -70.3(2) C14 C8 C1 C2 53.0(3) C7 C8 C1 C2 173.4(2) C9 C8 C1 C6 111.28(18) C14 C8 C1 C6 -125.39(17) C7 C8 C1 C6 -5.00(19) C6 C1 C2 C3 -0.9(3) C8 C1 C2 C3 -179.21(19) C4 C3 C2 C1 0.5(3) Cl1 C3 C2 C1 178.95(15) C9 C10 N2 O2 -0.7(2) C11 C10 N2 O2 179.71(19) O2 C12 C9 C10 -0.8(2) N3 C12 C9 C10 177.44(18) O2 C12 C9 C8 178.75(16) N3 C12 C9 C8 -3.0(3) N2 C10 C9 C12 1.0(2) C11 C10 C9 C12 -179.5(2) N2 C10 C9 C8 -178.5(2) C11 C10 C9 C8 1.0(4) C1 C8 C9 C12 127.5(2) C14 C8 C9 C12 1.0(2) C7 C8 C9 C12 -120.92(19) C1 C8 C9 C10 -53.1(3) C14 C8 C9 C10 -179.6(2) C7 C8 C9 C10 58.5(3) C9 C8 C14 C13 2.9(2) C1 C8 C14 C13 -123.2(2) C7 C8 C14 C13 122.75(19) C9 C8 C14 C15 -175.48(16) C1 C8 C14 C15 58.4(2) C7 C8 C14 C15 -55.6(2) C15 C14 C13 N3 173.17(17) C8 C14 C13 N3 -5.1(3) C15 C14 C13 C18 -6.8(3) C8 C14 C13 C18 174.89(17) O2 C12 N3 C13 179.11(16) C9 C12 N3 C13 1.0(3) C14 C13 N3 C12 3.1(3) C18 C13 N3 C12 -176.94(16) C14 C13 C18 C17 -22.5(3) N3 C13 C18 C17 157.52(17) C13 C18 C17 C20 -70.7(2) C13 C18 C17 C19 168.61(18) C13 C18 C17 C16 50.0(2) C20 C17 C16 C15 68.5(2) C19 C17 C16 C15 -171.06(18) C18 C17 C16 C15 -52.5(2) C13 C14 C15 O3 -173.34(18) C8 C14 C15 O3 5.1(3) C13 C14 C15 C16 4.5(3) C8 C14 C15 C16 -177.07(17) C17 C16 C15 O3 -155.17(19) C17 C16 C15 C14 27.0(3) O1 C7 N1 C6 175.33(18) C8 C7 N1 C6 -7.4(2) C5 C6 N1 C7 -174.1(2) C1 C6 N1 C7 4.2(2) C9 C12 O2 N2 0.4(2) N3 C12 O2 N2 -177.96(16) C10 N2 O2 C12 0.2(2)